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N-(3-aminopropyl)-3-{[1-(2-methyl-1,3-thiazol-4-yl)ethyl]sulfamoyl}benzamide
N-({1-[2-(naphthalen-1-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
2-[(3-methoxyphenyl)methyl]-8-(1H-pyrrole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-{2-oxo-2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}azepan-2-one
2-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-5-methoxyphenol
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(5-methylhexan-2-yl)-1,3-oxazole-4-carboxamide
4-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydroquinolin-2-one
(2S,4R)-N-ethyl-4-[2-(2-methylphenyl)acetamido]-1-(pent-4-enoyl)pyrrolidine-2-carboxamide
N-(2-hydroxyethyl)-3-[5-(pyridin-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
methyl 5-[(butan-2-yl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4-(dimethylamino)butanamide
9-{[2-(methylsulfanyl)phenyl]methyl}-3,9-diazaspiro[5.5]undecane-2,4-dione
3-(2-phenylethyl)-5-[4-(4H-1,2,4-triazol-4-yl)phenoxymethyl]-1,2,4-oxadiazole
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-3-ethyl-1H-pyrazole-5-carboxamide
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(furan-2-yl)-2-oxoacetamide
1-(2-ethoxyethyl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[methyl(piperidin-4-yl)amino]-1-[3-(3-methylphenoxymethyl)piperidin-1-yl]ethan-1-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[2-(2-methyl-1,3-thiazol-4-yl)acetamido]acetic acid
4-chloro-5-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
4-[4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
[3-(1H-imidazol-1-yl)propyl]({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
2-(2H-1,3-benzodioxol-5-yl)-8-methoxy-5-(quinolin-6-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
4-(2-methylquinolin-6-yl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidin-4-ol
3-[(4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)methyl]-2-methyl-1H-indole
1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-{[3-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(hydroxymethyl)piperidin-4-ol
6-({4-[4-(propan-2-yl)piperidine-1-carbonyl]-1,3-oxazol-2-yl}methoxy)quinoline
8-(2,2-dimethylcyclopropanecarbonyl)-3-[3-(4-ethylpiperazin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{2-[1-(2-ethoxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]piperidin-1-yl}-2-methoxyethan-1-one
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]acetamide
(3R,4R)-4-{[2-methyl-6-(trifluoromethyl)quinolin-4-yl]amino}piperidin-3-ol
4-benzyl-3-ethyl-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1,4-diazepan-5-one
2-{2-[(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-{2-[1-(2,6-difluoro-4-methoxybenzoyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
3-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[2-methyl-3-({[2-(methylsulfamoyl)ethyl]amino}methyl)-1H-indol-1-yl]acetamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(3-fluoro-4-methoxybenzoyl)pyrrolidin-3-yl]methanol
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(9H-purin-6-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(methoxymethyl)-6-methyl-4-oxo-1-(3-phenylpropyl)-N-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-6-phenylpyridazin-3-amine
1-(4-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperazin-1-yl)ethan-1-one
3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-[2-(propan-2-yl)phenyl]urea
N-[(2-{4-[3-(4-methoxyphenyl)propanamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]thiophene-3-carboxamide
5-(3-acetylphenoxymethyl)-N-[(3-fluorophenyl)methyl]-1H-pyrazole-3-carboxamide
4-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-(2-fluorophenyl)piperidine
3-(4-methoxyphenyl)-N-methyl-N-(oxan-4-yl)-3-phenylpropanamide
2-[(2,3-difluoro-4-methylphenyl)methyl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine