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N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
1-(2-methyloxane-2-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
1-{[2-(1-ethyl-1H-1,2,4-triazol-5-yl)-1H-imidazol-1-yl]methyl}cyclohexan-1-ol
N-(4-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}phenyl)ethane-1-sulfonamide
4-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-oxo-N-(propan-2-yl)-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
7-methyl-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-N-[1-(pyridin-3-yl)propyl]pyrimidin-2-amine
2-(5-methyl-1,2-oxazol-3-yl)-1-{[4-(trifluoromethoxy)phenyl]methyl}piperidine
N-(1-hydroxy-2-methylpropan-2-yl)-4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-(propan-2-yl)-4-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperazin-2-one
4-(1H-indole-5-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2,6-dimethylquinoline-4-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,4,6-trimethylpyrimidin-2-amine
2-(furan-2-yl)-5-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
5-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-2,1,3-benzothiadiazole
1-(1,3-dioxo-2-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-2,3-dihydro-1H-isoindol-4-yl)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)piperidine-3-carboxamide
N-{3-[methyl(phenyl)amino]propyl}-3-azaspiro[5.5]undecan-9-amine
1-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(1-cyclopentyl-1H-pyrazol-5-yl)urea
N-({1-[(3-phenoxyphenyl)methyl]piperidin-3-yl}methyl)furan-2-carboxamide
1-phenyl-4-[2-(phenylamino)pyrimidine-5-carbonyl]piperazin-2-one
4-(3-hydroxy-3-methylbutyl)-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
2-{2-[1-(1-methylpiperidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
(4S)-1-[(4-chloro-3-fluorophenyl)methyl]-3,3,4-trimethylpiperidin-4-ol
3-(2-ethyl-1H-imidazol-1-yl)-1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-cyclopropyl-2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]pyridine-4-carboxamide
1-(4-benzylpiperidin-1-yl)-3-[1-(oxane-4-carbonyl)piperidin-4-yl]propan-1-one
2-amino-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-4-methylpyrimidine-5-carboxamide
1-cyclopentanecarbonyl-N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]piperidine-4-carboxamide
3-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]-5-methyl-1H-indole-2-carboxylic acid
1-cyclopropyl-N-[2-(3-methylthiophen-2-yl)ethyl]-1H-pyrrole-2-carboxamide
3-(5-{[2-(furan-2-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)(1,3-thiazol-4-ylmethyl)amine
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
7-chloro-3-({methyl[2-(oxan-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
N-[4-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-2H-1,3-benzodioxole-5-carboxamide
4-(3-hydroxy-2-methylbenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
N-butyl-N-methyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-(2-hydroxy-2-methylpropyl)-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
(3S,4S)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4-propylpyrrolidine-3-carboxylic acid
5-methyl-1'-{[5-(oxan-2-yl)furan-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(3-fluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl]methanol
3-(2-methoxyethyl)-1-[3-(2-methoxyphenyl)propanoyl]piperidine-3-carboxylic acid
1-ethyl-4-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(3-phenoxypropanoyl)piperidin-4-yl]propanamide
1-cyclopentyl-5-(3-methylpiperidine-1-carbonyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide