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N-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-methylcyclopropane-1-carboxamide
3-(2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-4-(2-phenylethyl)piperazin-2-one
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl}){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
4-hydroxy-N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
N-(4-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenyl)acetamide
2-{6-[4-(ethanesulfonyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
butyl 4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
3-[4-(1H-imidazol-2-ylmethyl)piperazin-1-yl]-2,5-dimethylpyrazine
4-methyl-6-[3-(morpholin-4-ylmethyl)phenyl]pyrimidin-2-amine
N-[(1S)-1-cyclohexylethyl]-4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carboxamide
1-(4-{4-[4-(ethylamino)pyrimidin-2-yl]piperazin-1-yl}piperidin-1-yl)butan-1-one
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]acetamide
(1S,5R)-3-(6-aminopyridine-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[3-({[(3-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)-1H-indol-1-yl]acetamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-{3-[({2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}amino)methyl]-2-methyl-1H-indol-1-yl}acetamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
5-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
(3aR,5R,6S,7aS)-5,6-dihydroxy-N-(2,3,4-trifluorophenyl)-octahydro-1H-isoindole-2-carboxamide
7-chloro-N,3,5-trimethyl-N-[3-(1H-pyrazol-1-yl)propyl]-1-benzofuran-2-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
(3S,4R)-1-(3,6-dimethylpyrazin-2-yl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
1-[3-(2-methyl-4-phenylpiperazin-1-yl)-3-oxopropyl]azepan-2-one
3-amino-1-(7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
2-(3,4-dichlorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
(benzylsulfamoyl)[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]amine
(3aR,6aR)-2-methanesulfonyl-5-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-ethoxy-3-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N,2-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,6-naphthyridine-3-carboxamide
5-(1H-indol-1-ylmethyl)-N-methyl-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-3-carboxamide
2-{1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]pyrrolidin-2-yl}pyridine
2-(4-phenylpiperidin-1-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]acetamide
1-{1-[(3-methoxyphenyl)methyl]-5-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
1-(4-{[4-(3-chloropyridin-2-yl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
7-fluoro-2-methyl-N-[2-(N-methylmethanesulfonamido)ethyl]quinoline-4-carboxamide
2-(2-aminopyrimidin-5-yl)-N-cycloheptyl-N,8-dimethylquinoline-4-carboxamide
6-methyl-3-({methyl[1-(3-methylpyridin-2-yl)propan-2-yl]amino}methyl)-1,2-dihydroquinolin-2-one
4-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]pyridine
6-tert-butyl-N,1-dimethyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-[(2,3-dimethoxyphenyl)methyl]-2-[(6-methylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-({2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)ethyl]acetamide
(2S,4R)-4-amino-1-(5-methyl-2-phenylfuran-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(1,2,4-oxadiazol-3-ylmethyl)-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
3-(1-methyl-1H-1,3-benzodiazol-6-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]urea
4-[(3-methoxyphenyl)methyl]-1-[(5-methylthiophen-2-yl)methyl]-1,4-diazepan-5-one