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(3S,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(propan-2-yl)-3-({2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2-methylphenyl)methyl]piperidin-3-yl}propanamide
3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}-1-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]urea
1-(2-methoxy-5-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
(3S,9aR)-3-[(2S)-butan-2-yl]-8-[(5-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-1-(2-phenylethyl)-N-[(trimethylpyrazin-2-yl)methyl]piperidin-3-amine
(4aS,8aR)-1-(2-aminoethyl)-6-[(3-phenyl-1,2-oxazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
N-(2-methoxyethyl)-2,6-dimethyl-N-(1,3-thiazol-2-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide
(1S,5R)-6-(3-fluoro-4-methylbenzoyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2,3-dimethyl-6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoxaline
N-benzyl-N-methyl-3-[1-(4-oxo-4H-chromene-2-carbonyl)piperidin-4-yl]propanamide
5-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-2-methylpyrimidin-4-ol
1-cyclopentyl-4-(4-ethoxypyrimidin-2-yl)piperazin-2-one
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-(1H-pyrazol-4-yl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]butan-1-one
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-4-carboxamide
N-cyclopropyl-1-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[2-(4-methylpiperazin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[2-(2-chloro-4-fluorophenyl)-1H-imidazol-1-yl]butan-2-ol
4-[(2-chloro-6-fluorophenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]urea
3-(ethoxymethyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazole
4-({3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridine
2-[9-(cyclopentylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
1-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]-4-(4-methoxyphenyl)butane-1,4-dione
N-{3-[(2S)-2-amino-3-(1,3-thiazol-4-yl)propanamido]phenyl}-4-methylbenzamide
2-({3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
8-chloro-2-(furan-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]quinoline-4-carboxamide
4-{[3-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}quinoline
3-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
N-({5-[(3-fluoro-5-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-(2-methylphenyl)-3-phenylpropanamide
4-[1-(1-benzylpiperidin-4-yl)piperidin-3-yl]-5-(4-fluorophenyl)-2-methylpyrimidine
(4aS,8aS)-2-(3-chloropyridin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
2-[2-(pyridin-4-yl)ethyl]-9-(pyridine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(1H-pyrazol-4-yl)benzamide
N-{2-[1-(2-hydroxybutyl)-1H-1,2,4-triazol-5-yl]propan-2-yl}acetamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[1-(2-fluorophenyl)piperidin-4-yl]acetamide
4-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-methyl-3-phenyl-1H-pyrazole
4-(1-methyl-1H-pyrazole-3-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
N-cyclopentyl-1-methyl-5-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[2-({6-methylthieno[2,3-d]pyrimidin-4-yl}sulfanyl)acetyl]pyrrolidine-2-carboxamide
3-methyl-N-{2-[4-(1-methylpiperidin-4-yl)morpholin-2-yl]ethyl}furan-2-carboxamide
(3S,5S)-N-[(2,6-difluorophenyl)methyl]-1-(2,3-dihydro-1H-inden-2-yl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
1-{[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}azocane
5-[2-(2-ethylphenoxy)ethyl]pyridine-3-carboxamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide