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3,3-diphenyl-1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperidine
4-(3-chloro-2-fluorobenzoyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
8-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2-(2,4-difluorophenyl)ethyl]-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
2-(2-{2-[2-(thiophen-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}phenyl)ethan-1-ol
1-{6-[4-(pyridin-3-ylmethyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}azepane
methyl 4-({[(3S,5S)-1-[(2-chlorophenyl)methyl]-5-[(2-methoxyethyl)carbamoyl]pyrrolidin-3-yl]amino}methyl)benzoate
1-[2-(1H-imidazol-4-yl)acetyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
3-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}urea
(2E)-N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-3-(pyridin-3-yl)prop-2-enamide
N4-{2-[bis(propan-2-yl)amino]ethyl}-5-ethylpyrimidine-2,4-diamine
3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}urea
1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-4-(pyridin-2-yl)piperidin-4-ol
4-ethyl-3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[1-(3-methylbutanoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2,6-dimethoxy-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-3-carboxamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylsulfanyl)acetamide
2-(6-hydroxy-4-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-1,4-diazepan-1-yl)acetic acid
2-[methyl(5-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}pyrimidin-2-yl)amino]acetic acid
N-methyl-5-({3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
7-(morpholine-4-sulfonyl)-2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline
N-(furan-2-ylmethyl)-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[1-(2-hydroxyethyl)piperidin-4-yl]-1H-1,3-benzodiazole-2-carboxamide
2-{7-oxo-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-5-yl}benzoic acid
N,5,7-trimethyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
3-{imidazo[1,2-a]pyridin-2-yl}-N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]propanamide
(4aS,7aR)-N-(2-chlorophenyl)-4-(cyclopropylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-(1H-indol-4-ylmethyl)urea
3-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]-1-methyl-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]urea
N-(3-chloro-4-fluorophenyl)-3-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}propanamide
{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(trifluoromethyl)benzamide
N,N,1-trimethyl-3-(7-methyl-1H-indol-3-yl)-1H-1,2,4-triazol-5-amine
1-{2-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)ethyl]piperidin-1-yl}-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
5-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methylphenol
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine
(2S,4R)-1-[(2,5-dimethoxyphenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
N3-[(2-ethoxyphenyl)methyl]-N3-ethylpiperidine-1,3-dicarboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2-methoxyphenyl)methyl]piperidin-3-ol
4-(isoquinolin-5-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-({1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}amino)pyridine-3-carbonitrile
N-cycloheptyl-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-2,6-dioxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[4-(3-hydroxyphenyl)phenyl]-N-methylacetamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-{4-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamido]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-pyrrole-3-carboxamide
6-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-4-amine
8-[2-(trifluoromethoxy)benzenesulfonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(1-cyclohexylpiperidin-3-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide