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N-(5-oxo-1-propylpyrrolidin-3-yl)-2-(propan-2-yl)pyrimidine-4-carboxamide
4-(1-ethyl-1H-pyrazole-5-carbonyl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-3-amine
4-fluoro-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine
1-benzyl-5-(benzylamino)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-methyl-8-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3-phenyl-1,8-diazaspiro[4.5]decane
N5-cyclooctyl-N3-(2-methoxyethyl)-4-oxo-1-(oxolan-2-ylmethyl)-N3-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(2-{5-amino-4-cyano-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-trien-3-yl}phenoxy)propanoic acid
(1S,5R)-6-propyl-3-(quinoxaline-6-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-benzyl-1-(4,4,4-trifluorobutyl)pyrrolidin-2-one
8-[4-(3-hydroxy-3-methylbutyl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
4-({4-[3-(morpholin-4-yl)propoxy]phenyl}methyl)piperazin-2-one
3-[5-(2-propoxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
(1S,5R)-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2-methylpropyl)-8-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-cyclopropyl-1H-pyrazole-5-carboxamide
2-[(quinolin-6-yloxy)methyl]-N-[2-(1,3-thiazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)cyclohexanecarboxamide
6-oxo-1-(3-phenylpropyl)-N-[2-(1,3-thiazol-2-yl)ethyl]piperidine-3-carboxamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-2-ethylpyrimidine
2-methyl-7-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
N-[cyclopropyl(pyridin-2-yl)methyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
(3aR,6aR)-2-acetyl-5-{6,7,8,9-tetrahydro-5H-benzo[7]annulen-7-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[benzyl(methyl)amino]-2-{4-[(morpholine-4-carbonyl)amino]phenyl}acetic acid
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-[1-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-4-yl]-N,N-dimethylquinoline-4-carboxamide
3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-N-(isoquinolin-1-yl)benzamide
2-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
2-(2-hydroxynaphthalene-1-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(1-ethylpiperidin-3-yl)methyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
6-fluoro-4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
3-(2,5-difluorobenzoyl)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidine
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]acetamide
3-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
4-{4-[1-(2-chlorophenyl)-1H-1,2,4-triazol-5-yl]benzoyl}morpholine
(1S,5R)-6-(1H-imidazol-4-ylmethyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(4-methylphenyl)methyl]-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-methyl-5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
5-[({2-methoxy-5H,6H,7H-cyclopenta[b]pyridin-3-yl}formamido)methyl]thiophene-2-carboxylic acid
4-[2-(methylsulfanyl)pyridine-3-carbonyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
8-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-{4-[(2-hydroxy-7-methylquinolin-3-yl)methyl]piperazin-1-yl}pyrazine-2-carbonitrile
3-[1-(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-{2-[({4-[2-(3-methylpiperidin-1-yl)ethoxy]phenyl}methyl)amino]ethyl}piperidin-4-ol
8-[2-(diethylamino)acetyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{[2-(hydroxymethyl)-1H-1,3-benzodiazol-5-yl]formamido}-N,4-dimethylpentanamide
4-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(pyridin-2-ylmethyl)acetamide