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dimethyl({2-[4-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]phenyl}methyl)amine
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(2S,4S)-4-cyclobutaneamido-1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-N-ethylpyrrolidine-2-carboxamide
(2-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
6-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
9-(4-ethyl-5-methylthiophene-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 5-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)-N-(2-methoxyethyl)piperidine-3-carboxamide
5-[2-(morpholin-4-ylmethyl)phenyl]-2,3-dihydro-1λ6-thiophene-1,1-dione
3-phenyl-N-{1-[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
3-[(5-ethyl-2-methylpyrimidin-4-yl)amino]-1-(4-methylpiperidin-1-yl)propan-1-one
1-butyl-4-{[4-(2,2-dimethyloxan-4-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(thiophen-2-yl)propan-1-one
2-hydroxy-5-methoxy-N-{[1-(oxan-4-yl)piperidin-3-yl]methyl}benzamide
4-ethyl-1-methyl-3-{1-[(4-methylpiperazin-1-yl)sulfonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-hydroxyethyl)-9-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2-(3-methoxyphenyl)azetidine
N-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]cyclohexanecarboxamide
4,4-difluoro-1-({4-[2-(3-methylpiperidin-1-yl)ethoxy]phenyl}methyl)piperidine
methyl 2-(azepane-1-sulfonyl)-6-(2-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
6-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-N-ethylpyridine-3-carboxamide
2-methyl-N-[2-(morpholin-4-yl)ethyl]imidazo[1,2-a]pyrimidine-3-carboxamide
2-{4-[2-(4-propanamidophenoxy)acetyl]morpholin-3-yl}acetic acid
1-(2-cyclohexylethyl)-3-hydroxy-3-[(3-phenoxyazetidin-1-yl)methyl]piperidin-2-one
2-({[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)-N-(propan-2-yl)acetamide
5-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1-ethylpiperidin-2-one
{4-[({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]phenyl}methanol
5-(3-methoxyphenoxymethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
methyl[2-(oxan-4-yl)ethyl]{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(pyridin-3-yloxy)propyl]acetamide
(3S,4S)-4-cyclopropyl-1-[(1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)sulfonyl]pyrrolidine-3-carboxylic acid
2-methyl-4-phenyl-9-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane
(1S,5R)-3-[(3-hydroxyphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
5-methyl-2-[1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyridine-3-carboxamide
5-{1-[1-(benzenesulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyrimidine
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(oxolan-3-yl)benzamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazole
4-(3-hydroxybenzoyl)-1-(4-methoxyphenyl)piperazin-2-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[2-(diethylamino)acetyl]piperidine-4-carboxamide
5-{[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
3-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}pyridine
N-ethyl-6-[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxamide
1-methyl-6-(pyridin-3-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
dimethyl[(4-{1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-2-yl}phenyl)methyl]amine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
4-[(2-fluorophenyl)methyl]-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
(1R,5R)-6-(2-methoxyethyl)-3-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane