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2-methyl-5-(4-{[(thiolan-3-yl)amino]methyl}piperidin-1-yl)-2,3-dihydropyridazin-3-one
{3-[4-(2,6-dimethoxypyrimidin-4-yl)piperazin-1-yl]-2,2-dimethylpropyl}dimethylamine
(2R,3R,6R)-3-(4-fluorophenyl)-5-(pyridine-3-sulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{4-[(1-phenylethyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-5-methylthiophene-2-carboxamide
1-(4-methoxyphenyl)-4-[4-(1H-pyrazol-4-yl)butanoyl]piperazin-2-one
1-(3-chlorothiophene-2-carbonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-4-(4-methoxyphenyl)-4-oxobutanamide
2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-amine
(4-{6-[(dimethylamino)methyl]-1,4-oxazepane-4-carbonyl}phenyl)methanol
2-methyl-7-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[(2S)-oxolan-2-ylmethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 5-{[1-(dimethylamino)propan-2-yl]amino}-3-(furan-2-amido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{2-[1-(4-methoxybenzenesulfonyl)piperidin-2-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-(2-methoxyethyl)-1-[1-(2-phenylacetyl)piperidin-4-yl]piperidine-3-carboxamide
1-{6-[4-(morpholin-4-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}azepane
2-methyl-N-{1-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidine
1-benzyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,4-diazepan-6-ol
N,N-dimethyl-3-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]aniline
2-{[(3,5-dimethylphenyl)methyl]sulfanyl}-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
1'-(3,5,7-trimethyl-1H-indole-2-carbonyl)spiro[indene-1,4'-piperidine]
1-(2,2-dimethylpropyl)-3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-3-hydroxypiperidin-2-one
2-amino-N-{2-[cyclopentyl(methyl)amino]ethyl}-N,4-dimethylpyrimidine-5-carboxamide
5-(3-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,3,4-tetrazole
N-(2-methylpropyl)-1-[1-(1,3-thiazol-2-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
4-methyl-1-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}sulfonyl)piperidine
3,6-dimethyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-{3-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
6-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroquinoxaline-2,3-dione
5-(1H-indole-3-carbonyl)-1-methyl-N-[3-(morpholin-4-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3aR,6aR)-2-(3-cyclopropylpropanoyl)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-chloro-2-methoxybenzamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-(oxolane-2-carbonyl)piperidin-4-amine
3-[4-(1-hydroxy-3-methylbutyl)piperidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
2-[(2-ethylpyrimidin-5-yl)formamido]-4-(methylsulfanyl)butanoic acid
(2,2-diphenylethyl)(methyl)[2-(oxan-4-yl)ethyl]amine
2-(2-methoxyphenoxy)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
N-{4-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]-2-methoxyphenyl}acetamide
3,3-bis(2-methoxyethyl)-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}urea
2-[(1-carboxy-3-methylbutan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(3R,4R)-4-cyclobutyl-3-methyl-1-[2-(pyridin-2-yl)ethyl]piperidin-4-ol
(3S,4R)-N,N-dimethyl-1-(1-methyl-1H-pyrazole-4-carbonyl)-4-propylpyrrolidin-3-amine
N,N-diethyl-1-[(1s,4s)-4-[2-(pyridin-2-ylsulfanyl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrimidin-2-amine
8-[(6-methylpyridin-2-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-[({1-[(4-chlorophenyl)methyl]piperidin-3-yl}carbamoyl)methyl]-2-methylpropanamide
N-(cyclohex-1-en-1-ylmethyl)-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(3-chloro-2-fluorophenyl)pyridin-3-yl]cyclopropanecarboxamide
3-[(3R,4S)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol