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ethyl 5-(pyridine-4-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}propan-1-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]propanamide
N-(3-ethoxypropyl)-6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
7-(4-fluorophenyl)-2-[2-(pyrrolidin-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
5-methyl-N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)thiophene-2-carboxamide
3-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1-(3-methylcinnolin-5-yl)urea
8-{[4-(trifluoromethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
N-[(2-chlorophenyl)methyl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(prop-2-en-1-yl)benzamide
N-{2-[(4-fluorophenyl)formamido]ethyl}-3-(2-oxopiperidin-1-yl)propanamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methyl-N-(propan-2-yl)piperidine-3-carboxamide
5-[3-chloro-5-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-2-methoxypyridine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-methyl-3-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
5-{[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}-2-methoxyphenol
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-N,N-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl){[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}amine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-oxo-2H-chromene-3-carboxamide
(1R,5R)-3-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N4-[(1R,2R)-2-(benzyloxy)cyclopentyl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
3-{1-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-imidazol-2-yl}pyridine
2-methoxy-5-(3-methylthiophen-2-yl)pyridine
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazole
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
2-amino-4-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-thiazole-5-carboxamide
N-(3,4-dimethoxyphenyl)-5-[4-hydroxy-1-(thiophen-2-ylmethyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
[(2-chloro-5-ethoxy-4-propoxyphenyl)methyl]({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl})amine
2-hydroxy-1-[4-(4-methylphenoxy)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
(cyclobutylmethyl)({4-[4-(furan-2-carbonyl)piperazin-1-yl]quinazolin-2-yl}methyl)(oxolan-2-ylmethyl)amine
7-methyl-N-(naphthalen-1-yl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
4-[2-(1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperidin-2-yl)ethyl]phenol
(1S,4S)-5-(2-amino-6-methylpyrimidin-4-yl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-{[2-(diethylamino)pyridin-3-yl]methyl}-1-(3-methoxyphenyl)urea
3-methyl-8-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(4-methoxyphenyl)ethyl]-5-(3-methyl-1H-pyrazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-(1H-1,2,3-benzotriazol-5-yl)-1-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]urea
3-{1-[2-methyl-3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-2-oxo-8-(1-phenylcyclopropanecarbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]isoquinoline
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
1-[1-(5-cyanopyridin-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
1-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
N-methyl-5-{[methyl(2-phenylethyl)amino]methyl}-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
(3S)-3-benzyl-4-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperazin-2-one
4-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-2-methylphenol
N-[2-(cyclohexylsulfanyl)ethyl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanamide
2-ethoxy-5-[2-({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)pyrimidin-4-yl]benzoic acid
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(propan-2-yl)-1H-pyrazole-4-carboxamide