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(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-N5-[2-(1H-imidazol-4-yl)ethyl]piperidine-3,5-dicarboxamide
N'-cycloheptyl-N-(1-hydroxyhexan-2-yl)butanediamide
1-{2-[1-(2-{[(2-fluorophenyl)methyl](methyl)amino}acetyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-9H-fluorene-9-carboxamide
3-(3-fluorophenyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-3-cyclohexyl-1H-pyrazole-4-carboxamide
N-methyl-3-{1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperidin-3-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
N-(5-hydroxyadamantan-2-yl)-4-{[2-(4-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(2S)-1-hydroxy-4-methylpentan-2-yl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
ethyl 4-(4-{2-[(4-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperazin-1-yl)piperidine-1-carboxylate
(4aS,7aR)-N-(3,4-dimethoxyphenyl)-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(3S,4R)-3-benzyl-N-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-methylpiperidin-4-amine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(2-fluorophenyl)methyl]-3-(3-methoxyphenyl)-N-propyl-1H-pyrazole-4-carboxamide
ethyl 4-[4-(6-chloropyridazin-3-yl)piperazin-1-yl]piperidine-1-carboxylate
2-(4-fluorophenyl)-N-(3,4,5-trimethoxyphenyl)azetidine-1-carboxamide
1-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
2-(4-fluorophenoxy)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(pyridin-4-yl)piperazine
5-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
3-{1-[2-(4-fluorophenyl)benzoyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
(1R,3S,5S)-8-({3-ethoxy-4-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-8-azabicyclo[3.2.1]octan-3-ol
8-(1H-1,3-benzodiazol-2-ylmethyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
(3S,4S)-1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
methyl(piperidin-3-ylmethyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
1,3-dimethyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-(5-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}furan-2-yl)-1H-pyrazole
1-{1'-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4-(4-methylphenoxy)piperidine
5-[5-(oxolan-2-yl)thiophen-2-yl]-3-(2-phenylethyl)-1H-1,2,4-triazole
6-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5,6-dihydro-1,6-naphthyridin-5-one
N-cyclohexyl-4-(5-{[(2-methoxyphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidine-1-carboxamide
5-(5-fluoro-2-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
[1,3-bis(2-phenylethyl)piperidin-3-yl]methanol
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-propyl-1,3-thiazole-4-carboxamide
N-(1-cyclopentyl-1H-pyrazol-5-yl)-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-3-methyl-1-(3-methylcinnolin-5-yl)urea
2-amino-4-[2-methoxy-5-oxo-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
2-[9-(1-methyl-1H-pyrrole-2-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-(4-{4-[(oxolan-2-ylmethyl)amino]piperidin-1-yl}phenyl)-3-phenylpropanamide
methyl[1-(3-methylpyridin-2-yl)propan-2-yl](quinolin-4-ylmethyl)amine
1-(2-hydroxyethyl)-N-[(3-phenylphenyl)methyl]piperidine-3-carboxamide
(1S,5R)-3-(4-fluoro-2-methylbenzenesulfonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-(2-fluorophenyl)propyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
5-methanesulfonyl-N-[2-(piperidin-1-yl)ethyl]-4-(piperidin-3-yl)pyrimidin-2-amine
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,2,4-triazol-3-yl]acetamide
5-[1-(4-methoxyphenyl)cyclopentyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole