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1-(5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
(4aR,7aS)-1-[(3,5-dimethylphenyl)methyl]-4-(1H-imidazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-1-phenylpiperazin-2-one
N-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethylpiperidin-4-amine
1-(4-methylpiperazin-1-yl)-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propan-1-one
3-(azocan-1-yl)-N-[2-(methylsulfamoyl)ethyl]propanamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-5-propyl-1,2-oxazole-4-carboxamide
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-[2-(cyclohexylsulfanyl)ethyl]-4-(1H-pyrazol-4-yl)butanamide
1-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)-3-(1H-pyrazol-4-yl)propan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[(1-methyl-1H-imidazol-5-yl)methyl]piperazin-2-one
4-cyano-N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1-methyl-1H-pyrrole-2-carboxamide
3-(3-hydroxyphenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
1'-(pyridin-4-ylmethyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
methyl (2S,4R)-1-methyl-4-[3-(1H-1,2,4-triazol-1-yl)propanamido]pyrrolidine-2-carboxylate
1-{4-[1-(2,3-dimethylphenyl)piperidin-4-yl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
2,3,6-trimethyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)quinoline-4-carboxamide
N-methyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(oxolan-3-yl)piperidine-4-carboxamide
N3-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-N5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-[4-(pyridin-3-yloxy)phenyl]urea
N-ethyl-2-(4-hydroxypiperidin-1-yl)-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)acetamide
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-(morpholin-3-yl)ethan-1-one
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-(oxan-4-yl)ethan-1-one
2-[(3S,4R)-3-cyclopropyl-4-[2-(ethylamino)-4-methyl-1,3-thiazole-5-amido]pyrrolidin-1-yl]acetic acid
({4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-5-phenylfuran-2-yl}methyl)diethylamine
1-ethyl-8-(furan-3-ylmethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(2-{[(2-methoxyphenyl)methyl]carbamoyl}ethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-4-yl}thiomorpholine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}benzamide
2-[1-(3-phenylpropyl)pyrrolidin-3-yl]acetic acid
(4aS,8aR)-6-(3-fluorobenzenesulfonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-1-cyclopropyl-N-methyl-5-oxopyrrolidine-3-carboxamide
[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N-[(1-ethylpyrrolidin-2-yl)methyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-({[2-methyl-6-(propan-2-yl)phenyl]carbamoyl}methyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
2-{[(1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)oxy]methyl}pyridine
1-[4-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
2-(3-hydroxypropyl)-9-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-amino-4-(pyridin-3-yl)-6-(2,4,5-trifluorophenyl)pyridine-3-carbonitrile
N-(2-fluoro-4-methoxyphenyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carboxamide
1-(2-ethoxypyridine-3-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-(azocan-1-yl)-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylacetamide
2-ethyl-4-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}pyrimidine
1-cyclopropyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxamide
4-{[4-(2-aminopyrimidin-4-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
[1-({1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
N3-(5,6-dimethylpyrimidin-4-yl)-N1-(pyridin-3-yl)propane-1,3-diamine
[(3R,4R)-1-[1-(3-chlorophenyl)piperidin-4-yl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1,3-dimethyl-5-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}imidazolidine-2,4-dione