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1-[(6-hydroxypyrimidin-4-yl)methyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
(4aR,7aS)-1-cyclopropanecarbonyl-4-(1H-imidazol-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,5S)-N3-[2-(1H-imidazol-1-yl)ethyl]-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
(2S)-1-{4-phenyl-5-[4-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}propan-2-ol
7-(cyclohexylmethyl)-2-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
8-(1H-indol-3-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{2-[3-(3-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}-3-propylimidazolidine-2,4-dione
3-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
(1S,5R)-3-cyclobutanecarbonyl-6-(2-methylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2,5-dioxoimidazolidin-1-yl)-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]acetamide
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]pyridine-3-carboxamide
2-(5-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
6-[2-(tert-butylsulfamoyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-{[4-(methylsulfanyl)phenyl]methyl}-4-oxo-N-propyl-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-{1-[1-(4-methoxy-3,5-dimethylbenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-1-(propan-2-yl)piperidine-3-carboxamide
1-[3-(4-chlorobenzoyl)piperidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
3,7-dimethyl-8-(1-methyl-1H-pyrazol-4-yl)-2,3,6,7-tetrahydro-1H-purine-2,6-dione
1-cyclopentyl-4-({[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}methyl)pyrrolidin-2-one
1-ethyl-N,3-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-3-carboxamide
5-[4-(benzyloxy)-4-(prop-2-en-1-yl)piperidine-1-carbonyl]-2-methylpyrimidin-4-ol
9-[(4-ethylphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(6-methyl-2-phenyl-1,2-diazinane-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
1-methyl-4-(3-propoxypiperidin-1-yl)piperidine
1-(4-methoxybenzenesulfonyl)-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazine
1-{5-methyl-6-[2-(pyridin-3-yl)piperidine-1-carbonyl]thieno[2,3-d]pyrimidin-4-yl}azepane
5-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
N-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}propanamide
6-{2-[2-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-imidazol-1-yl]ethyl}-2-methylpyrimidin-4-ol
6-ethyl-2-methyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]quinoline-4-carboxamide
N-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-[3-(trifluoromethyl)phenyl]acetamide
(3S,4R)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-{1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}ethan-1-ol
3-(4-chloro-1H-pyrazol-1-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
5-methyl-3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-indazole
4-[3-(1,3-benzothiazol-2-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(5-methylpyrazin-2-yl)methyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
2-amino-2-methyl-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
4-(4-cyclobutyl-6-methylpyrimidin-2-yl)piperazine-1-sulfonamide
2-(2-methoxy-4-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}phenoxy)acetamide
(furan-3-ylmethyl)(methyl){[(2R,5S)-5-(pyridin-3-ylmethyl)oxolan-2-yl]methyl}amine
N-cyclopentyl-5-(1H-imidazole-4-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-[(propan-2-yl)amino]pyridine-3-carboxamide
1-propyl-N-(pyridin-4-ylmethyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(1H-imidazol-1-yl)propyl]-2,8-dimethylquinoline-4-carboxamide