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(2S,4R)-4-amino-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]-N-methylpyrrolidine-2-carboxamide
N-methyl-5-(morpholin-4-ylmethyl)-N-[2-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
3-(5-{[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
(4aS,8aR)-6-[5-(methoxymethyl)furan-2-carbonyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
5-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-2-(pyrrolidin-1-yl)pyrimidine
N-{5-[3-(5-chloro-2-hydroxyphenyl)-1H-pyrazol-1-yl]pyridin-2-yl}acetamide
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-[3-(dimethylamino)propyl]-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-3-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}piperidine
2-[({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)amino]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
7-chloro-3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3,4-dihydroquinazolin-4-one
methyl 6-(cyclopent-1-ene-1-carbonyl)-2-{[2-(4-fluorophenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}pyridine-3-carbonitrile
1-[(2,3-difluorophenyl)methyl]-3-(3-methoxyphenoxy)azetidine
1-[6-(6-methoxypyridin-3-yl)pyridine-3-carbonyl]-4-phenylazepane
methyl[(3-methylpyridin-4-yl)methyl][(2-phenyl-1,3-oxazol-4-yl)methyl]amine
4-[1-cyclohexyl-3-(ethoxymethyl)-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
3-[3-(phenoxymethyl)-5-(pyrazin-2-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
(1S,4S)-2-(3-chlorophenyl)-5-[(1-methyl-1H-pyrrol-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
4-(1H-1,3-benzodiazol-1-yl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
3-[(2R,3R,6R)-5-(5-ethyl-2-methylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(pyrrolidin-1-yl)benzamide
N-cyclobutyl-2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
8-(cyclopropylmethyl)-N-[(4-methoxyphenyl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
3-[(3-cyclopentyl-1,2,4-oxadiazol-5-yl)methyl]-2,3-dihydro-1H-isoindol-1-one
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(4-methylphenyl)propyl]-1,3-oxazole-4-carboxamide
methyl 6-[(2-ethoxyphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
[(2-methoxyphenyl)methyl](prop-2-en-1-yl)(quinolin-2-ylmethyl)amine
(2R,3R,6R)-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)-3-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]urea
2-amino-N-(cyclohex-1-en-1-ylmethyl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
[(3R,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-4-(2-methylphenyl)piperazine
2-methyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
6-(4-ethylpiperazin-1-yl)-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-(2-hydroxy-4-methoxybenzoyl)pyrrolidine-3-carboxylic acid
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
N-{4-[2-(4-hydroxyphenyl)acetamido]phenyl}-5-methylfuran-2-carboxamide
N-[2-(benzyloxy)ethyl]-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(methylamino)ethan-1-one
2-({6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(1H-imidazol-2-yl)benzamide
4-hydroxy-N-[3-(1H-indol-1-yl)propyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
[3-methyl-9-(quinolin-4-yl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
1-[(3-methoxyphenyl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(pyridine-2-carbonyl)piperidin-4-amine
N-{1-oxaspiro[4.5]decan-3-yl}-3-propyl-1H-pyrazole-5-carboxamide
N-[(5-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
2-[3-(2-fluorophenyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
7-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,7-diazaspiro[4.5]decane