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2-[(3-chlorophenyl)methyl]-N-(oxan-4-ylmethyl)-1,3-benzoxazole-6-carboxamide
5-cyclobutanecarbonyl-1'-[(3-methylpyrazin-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
5-(1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,2,3-triazol-4-yl)-N-(propan-2-yl)pyrimidin-2-amine
4-(difluoromethoxy)-N-ethyl-N-(1-hydroxypropan-2-yl)benzamide
N-[3-(4-fluorophenyl)phenyl]-1-propanoylpyrrolidine-2-carboxamide
(3R,4S)-4-propyl-1-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]pyrrolidin-3-amine
1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-[(3-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
3-[2-(4-fluorophenyl)ethyl]-1-(1H-pyrazole-3-carbonyl)piperidine
5-oxo-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyrrolidine-3-carboxylic acid
1-(1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-1-oxopropan-2-yl)pyrrolidin-2-one
2-(dimethylamino)-2-(2-methylphenyl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
5-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-3-methyl-1,2-oxazole
4-{[2-(2-oxoimidazolidin-1-yl)ethyl]amino}-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
N,5-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-oxazole-4-carboxamide
2-(3-hydroxypropyl)-8-(1H-indole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(2-methyl-1H-imidazol-1-yl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]butan-1-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-(4-methylpyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-3-(2,1,3-benzothiadiazol-5-ylmethyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3,5-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1-benzofuran-2-carboxamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
3-[(4-methoxyphenyl)methyl]-1-methyl-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-cyclopropyl-1-(6-methylpyridin-3-yl)-3-[(3-methylthiophen-2-yl)methyl]urea
(3S,4S)-4-cyclopropyl-1-(6-cyclopropylpyrimidin-4-yl)pyrrolidine-3-carboxylic acid
1-[2-(1H-imidazol-5-yl)ethyl]-5-(oxan-4-yl)-3-phenyl-1H-1,2,4-triazole
3-[(3R,4S)-1-[(1-methyl-1H-indol-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
(1R,9aR)-1-{[(3-methoxypropyl)(1-methylpiperidin-4-yl)amino]methyl}-octahydro-1H-quinolizin-1-ol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-[2-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-6-methoxyphenoxy)ethyl]-1H-imidazole
2-(dimethylamino)-1-[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]-2-(3-fluorophenyl)ethan-1-one
N3-cyclohexyl-1-(2-methylpropyl)-4-oxo-N5-[2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxylate
4-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
4-methoxy-N-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
methyl 1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidine-2-carboxylate
4-hydroxy-2-(4-methylphenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide
N-(pyridin-2-ylmethyl)-3-{[1-(thian-4-yl)piperidin-4-yl]oxy}benzamide
2-amino-4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
2-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[1-(pyrazin-2-yl)propan-2-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
ethyl 4-oxo-1-pentyl-5-phenoxy-1,4-dihydropyridine-3-carboxylate
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-5,6-dimethyl-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-{4-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]piperidin-1-yl}ethan-1-one
1-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-3-(4-methoxyphenyl)propan-1-one
1-(4-benzylpiperazin-1-yl)-3-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl}propan-1-one
4-ethyl-3-({1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-(4-methyl-1,3-thiazole-5-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
methyl (2S,4R)-4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidine-2-carboxylate