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4-(2-methoxyphenyl)-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidine
(3S,4S)-1-[(3-cyanophenyl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
ethyl 1-({7-fluoro-2-oxo-1-[2-(piperidin-1-yl)ethyl]-1,2-dihydroquinolin-3-yl}methyl)piperidine-4-carboxylate
(3R)-1-({1-[1-(5-propylpyrimidin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-amine
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[3-(4-fluorophenyl)pyrrolidin-1-yl]ethan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2R,3R,6R)-5-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]methyl}-1H-pyrazole
3-[({1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]piperidin-4-yl}oxy)methyl]pyridine
2-(dimethylamino)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-2-(2-methylphenyl)acetamide
2-methyl-1-{2-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1H-indole-3-carbonitrile
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-(2-chloro-4-fluoro-5-methylphenyl)-2-(morpholin-4-ylmethyl)piperidine-1-carboxamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]butan-1-one
(3R,4S)-4-propyl-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-3-(4-methylpiperazin-1-yl)propan-1-one
1-{[2-(difluoromethoxy)phenyl]methyl}-4-(oxan-4-yl)piperazine
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-N-(2,4-dimethylphenyl)piperidine-1-carboxamide
1-{[(2S,4S)-1-(4-chloro-2-hydroxybenzoyl)-4-fluoropyrrolidin-2-yl]methyl}-3,3-diethylurea
2-methyl-6-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
2-{1-[(4-ethoxyphenyl)methyl]-4-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
8-(3,4-dimethylbenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1R,3S)-3-(2-hydroxyethoxy)-7-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
3-(4-methyl-1,3-thiazol-5-yl)-1-{4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
(2H-1,3-benzodioxol-4-ylmethyl)(methyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
3-{[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]methyl}-1λ6-thiane-1,1-dione
N-cyclopentyl-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-{1-[(3,4-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(2-methoxyphenyl)-1-benzofuran-2-carboxamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
9-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-(cyclopentylmethyl)-N,6-dimethyl-4-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(3S,4S)-4-(4-fluorophenyl)-1-(quinolin-8-ylmethyl)piperidin-3-ol
4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-(1,2-oxazol-5-yl)phenol
6-[4-(2-hydroxyethyl)piperidin-1-yl]-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
N,N-dimethyl-1-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-amine
2-(1,3-benzoxazol-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
6-(2,5-dimethylfuran-3-yl)-2-(2-methylpyrrolidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
(7R,9aR)-N-(3-fluorophenyl)-7-[(1S)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-methyl-N-(2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)methanesulfonamide
2-cyclopropyl-8-[(4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-methyl-2-[3-(morpholin-4-ylmethyl)phenyl]pyrimidin-4-amine
1-[(2-fluorophenyl)methyl]-4-[3-(2-methoxyphenyl)propanoyl]piperazin-2-one
1-[(2,4-dimethoxyphenyl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
5-(2-benzyl-1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3,3-dimethyl-1-(2-oxo-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethyl)urea
8-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
1-[2-(1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one