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(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]piperidin-4-ol
8-(benzenesulfonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-{2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
1-cyclohexyl-N3-cyclopropyl-4-oxo-N5-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1,2-dimethyl-N-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}-1H-imidazole-4-sulfonamide
N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-2-[4-(6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]acetamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
2-(2-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenoxy)ethan-1-ol
N-methyl-6-(2-methylpropyl)-2-oxo-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-dihydropyrimidine-4-carboxamide
4-(naphthalen-2-yloxy)-1-(quinolin-2-yl)piperidine-4-carboxylic acid
4-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}-1,4-diazepan-2-one
4-benzyl-4-(hydroxymethyl)-N-(2-phenylphenyl)piperidine-1-carboxamide
2-{[2-(dimethylamino)ethyl](methyl)amino}-N-(2-methylpropyl)-6-[4-(methylsulfanyl)phenyl]pyridine-3-carboxamide
6-{[butyl(methyl)amino]methyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(6-hydroxy-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1,4-diazepan-1-yl)-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
3-(cyclopropylmethyl)-1-[(8-methoxyquinolin-2-yl)methyl]piperidine-3-carboxylic acid
5-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-4-(piperidin-3-yl)benzamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole-6-carboxamide
3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-N-(1,3-thiazol-2-yl)benzamide
N-(cyclohexylmethyl)-3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
4-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)oxane-4-carbonitrile
(3R,4R)-3,4-dimethyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-ol
(2S)-2-{[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}-4-methylpentanamide
5-(oxolan-2-yl)-3-(4H-1,2,4-triazol-4-ylmethyl)-1,2,4-oxadiazole
1-(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)piperidine-4-carboxamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-methyl-1,2,3,6-tetrahydropyridine
2-(2,5-dimethylphenyl)-5-(methanesulfonylmethyl)pyridine
[(3R,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
2-[1-(6-cyclopropylpyrimidin-4-yl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
N,8-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-{3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}ethan-1-one
1-[(4-chlorophenyl)methyl]-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
[(3-{2-[4-(2H-1,3-benzodioxole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
[(4-fluorophenyl)methyl]({[2-(propan-2-yl)pyrimidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
4-{[4-(2-methyl-5-propylpyrimidin-4-yl)piperazin-1-yl]methyl}benzoic acid
N-[2-(ethylsulfanyl)ethyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
[1-(furan-3-carbonyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
4-methyl-5-{1-[3-(6-methylpyridin-2-yl)propyl]-1H-pyrazol-3-yl}-N-[(2,4,5-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
7-(cyclobutylmethyl)-2-[3-(furan-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(5-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
ethyl 3-[(2-fluorophenyl)methyl]-1-[3-(pyridin-3-yl)propanoyl]piperidine-3-carboxylate
4-[2-(1H-imidazol-4-yl)acetyl]-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
2-cyclopropyl-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyrimidine-5-carboxamide
4-ethyl-3-{[1-(quinoxaline-5-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
{2-oxo-2-[7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethyl}urea
2-(furan-2-yl)-1-(propane-1-sulfonyl)azepane
7-(2,3-dimethoxybenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
diethyl({2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine