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N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1-(2-phenylethyl)piperidin-4-amine
ethyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amine
2-(6-methoxypyridin-3-yl)-4-(piperidine-1-carbonyl)pyridine
5-{4-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-(3,4-dichlorophenyl)-4-(2-propylpyridine-4-carbonyl)morpholine
1-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
3-(1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methoxyphenyl)urea
1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-[(4-fluorophenyl)methyl]-1,4-diazepane
1-{[2-(furan-2-yl)phenyl]methyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
6-(4-hydroxypiperidin-1-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
N,N-diethyl-2-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoacetamide
8-(3,6-dimethylpyrazin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
dimethyl(2-{4-[2-(methylsulfanyl)benzoyl]morpholin-2-yl}ethyl)amine
(3S,4R)-1-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
[3-(1H-1,3-benzodiazol-2-yl)propyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
5-(2-methylpropyl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,2-oxazole-3-carboxamide
(3aR,7aS)-5-methyl-2-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-{[1-(dimethylamino)cyclohexyl]methyl}benzamide
methyl 4-(5-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
6-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexane-3-carbonyl]pyridin-2-amine
3-{1-[2-(6-methylpyridin-2-yl)ethyl]piperidin-3-yl}benzoic acid
8-cyclopropanecarbonyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-methyl-N-({1-[(2E)-2-methylpent-2-en-1-yl]piperidin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]pyrrolidin-2-one
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethylacetamide
4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-1-methyl-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
1-(5-aminopentanoyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
4-(2-methoxyphenoxy)-1-(pyridin-3-ylmethyl)piperidine-4-carboxylic acid
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)piperidin-2-one
4-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-1,4-diazepan-2-one
(2H-1,3-benzodioxol-4-ylmethyl)(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
1-(1-benzofuran-2-ylmethyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
2-[1-(3-benzyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidin-3-yl]-1,3-benzoxazole
6-{2-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}-1H-indazole
6-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}pyridine-3-carboxylic acid
(2S,4S)-N-ethyl-1-(1,3-thiazol-2-ylmethyl)-4-(thiophene-3-amido)pyrrolidine-2-carboxamide
1-(5-methyl-1,3,4-oxadiazol-2-yl)-3-[2-(methylsulfanyl)benzoyl]piperidine
1-(furan-3-ylmethyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-({[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}amino)-1-phenylpyrrolidin-2-one
1-[2-(dimethylamino)-6-(1H-pyrrole-2-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
8-(6-methylpyridazin-3-yl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(2-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrrol-1-yl)pyridine
1-[2-fluoro-3-(trifluoromethyl)phenyl]-3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
5-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]-2-(thiophen-2-yl)pyrimidin-4-ol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-ethyl-N-[2-(phenylsulfanyl)ethyl]acetamide
3-cyano-5-fluoro-N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}benzamide