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[1-(2-methoxy-5-methylbenzenesulfonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
2-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-1,3-thiazole-4-carboxamide
1-[2-methoxy-5-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
(2S,4R)-4-amino-N-ethyl-1-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)pyrrolidine-2-carboxamide
1-cyclohexyl-N3-[(2,4-dimethoxyphenyl)methyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[4-(1-methoxyethyl)phenyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridine
3,6-dimethyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-methoxyphenyl)acetamide
N-(2,3-dihydro-1-benzofuran-3-yl)-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
3-(3-fluorophenyl)-3-{2-[3-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
2-methyl-4-{4-[3-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]phenyl}butan-2-ol
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-(oxan-4-yl)-2-phenylacetamide
1-{3-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]phenyl}ethan-1-one
3-(2-methylpiperidin-1-yl)-N-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]azetidine-1-carboxamide
N-cyclopropyl-1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]piperazine-2-carboxamide
5-fluoro-6-methyl-2-(3-{[(prop-2-en-1-yl)(pyridin-3-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
2-[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carboxylic acid
1-(cyclohexylmethyl)-5-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]piperidin-2-one
(5-{1-[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]-1H-imidazol-2-yl}furan-2-yl)methanol
2-(4-methoxyphenyl)-N-{[1-(pyridazine-4-carbonyl)piperidin-3-yl]methyl}acetamide
2-{[2-(3-methyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]methyl}-1,3-thiazole
N-[(2-chlorophenyl)methyl]-3-[1-(1H-imidazole-4-carbonyl)piperidin-3-yl]propanamide
(1R,3S)-3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]cyclopentan-1-amine
1-[(4aR,8aR)-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridin-1-yl]-2-(2,6-difluorophenyl)ethan-1-one
N-ethyl-5-(1H-indol-1-ylmethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
3-ethyl-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-5-methyl-1,2-oxazole-4-carboxamide
1-[6-({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amino)pyridin-3-yl]ethan-1-one
1-[4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]piperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
N-benzyl-3-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-(2-phenylethynyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(isoquinoline-5-carbonyl)-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
N-(2-{[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-yl]formamido}ethyl)pyridine-3-carboxamide
1-[(1R)-1-(4-fluorophenyl)ethyl]-3-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]benzonitrile
N-[1-(pyrazin-2-yl)propan-2-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
(2S,4R)-1-benzyl-N-[2-(2-fluorophenyl)ethyl]-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
(3S,4S)-1-[2-(prop-2-en-1-yloxy)benzoyl]piperidine-3,4-diol
N,4-dimethyl-N-[3-(4-methylphenoxy)propyl]-3-(2-oxoimidazolidin-1-yl)benzamide
1-(diphenylmethyl)-N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-1H-1,2,3-triazole-4-carboxamide
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
5-ethyl-4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,6-dimethylpyrimidine
2-methyl-N-[3-(3-oxopiperazin-1-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
2-(2-hydroxyethyl)-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(3R,4S)-1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-3,4-dimethylpiperidin-4-ol
1-[3-(benzyloxy)phenyl]-3-[(1-methylpiperidin-2-yl)methyl]urea
1-(3-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
(3R,4R)-4-ethyl-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidine-3,4-diol
4-{5-[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]-4-phenyl-1H-imidazol-1-yl}butan-2-ol
methyl 4-{[4-(benzenesulfonyl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate