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N-[2-(adamantan-1-yl)ethyl]-N-methyl-1,1-dioxo-1λ6-thiane-4-carboxamide
5-(morpholin-4-ylmethyl)-N-[(1R,2S)-2-phenylcyclohexyl]furan-3-carboxamide
4-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-3-methyl-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
4-{2-azaspiro[4.4]nonane-2-carbonyl}-3,6-dimethyl-2-(1H-pyrazol-4-yl)quinoline
1-[3-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
[(2-ethylpyrimidin-5-yl)methyl](methyl){[3-(methylsulfanyl)phenyl]methyl}amine
7-[(3,4-difluorophenyl)methyl]-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
1-propyl-N-[2-(pyridin-4-yl)ethyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-amino-6-(4-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}piperazin-1-yl)pyrimidin-4-ol
3-fluoro-2-(2-fluoro-5-methoxyphenyl)pyridine
1-cyclopentyl-N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
(2E)-1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-3-(pyridin-2-yl)prop-2-en-1-one
8-(1H-indol-2-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
{1-[4-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
[2-(2,6-dimethylphenoxy)ethyl](ethyl)(pyridin-2-ylmethyl)amine
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-yl}-1H-1,2,4-triazole
ethyl 1-(cyclopropylmethyl)-5-(1H-pyrazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[3-(3-chlorophenyl)-N-methyl-3-phenylpropanamido]-N-methylpropanamide
ethyl 2-(4-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}morpholin-3-yl)acetate
2-[(1S,5R)-3-[(4-acetamidophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine
1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-5-phenyl-1H-pyrrole-2-carboxamide
N-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
N-{[7-fluoro-2-(thiophen-3-yl)quinolin-3-yl]methyl}cyclopropanamine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-[(3-methylpyridin-2-yl)methyl]-4-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperazine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-N'-[2-(propan-2-yl)phenyl]butanediamide
1-(2-methoxy-4-{[methyl(thian-4-yl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
N-(2-methoxyethyl)-4-methyl-3-{[(pyridin-3-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-(morpholin-4-ylmethyl)-N-[phenyl(pyridin-4-yl)methyl]-1,2-oxazole-3-carboxamide
N-cyclohexyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)butanamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-{4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]morpholin-3-yl}acetamide
5-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-decahydro-1,6-naphthyridin-2-one
5-(2-ethylphenyl)-1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazole
2-(4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}morpholin-3-yl)-1-(pyrrolidin-1-yl)ethan-1-one
2-(2-chloro-6-methoxyphenyl)-2-(thiomorpholin-4-yl)acetic acid
(3R,4R)-4-ethyl-1-(4-methoxyquinoline-2-carbonyl)piperidine-3,4-diol
4-(1-{3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]propanoyl}piperidin-3-yl)benzoic acid
1-cyclohexyl-N,N-bis(prop-2-en-1-yl)-1H-1,2,3-triazole-4-carboxamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}propan-1-one
N-(5-methyl-1,2-oxazol-3-yl)-2-oxo-2-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]acetamide
2-[1-(2-fluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]morpholine
4-(1-butyl-1H-imidazol-2-yl)-1-(1-phenylcyclopropanecarbonyl)piperidine
3-(4-methylphenyl)-3-phenyl-1-[3-(1H-pyrazol-1-yl)azetidin-1-yl]propan-1-one
1-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-4-yl}-3-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-methylurea
2-methyl-4-(3-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}phenyl)butan-2-ol
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[2-(furan-2-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol