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5-(3-acetylphenoxymethyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1R)-1-phenylethyl]urea
1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
N-[4-(propan-2-yl)phenyl]-1-(1H-pyrazol-3-ylmethyl)piperidin-3-amine
methyl[(6-methylpyridin-2-yl)methyl]{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
1-{4-[3-(phenylamino)piperidin-1-yl]piperidin-1-yl}ethan-1-one
1-[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
1-(4-methylpiperazin-1-yl)-3-(4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}phenoxy)propan-2-ol
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2,6-dimethylbenzamide
2-ethyl-4-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1-(propan-2-yl)piperazine
2-(3-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}phenyl)ethan-1-amine
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]propan-2-ol
2-cyclopropyl-9-(2-ethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 5-[(cyclopropylamino)methyl]-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-pyrazole-4-carboxylate
2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-6-methoxy-1-methyl-1H-indole
N,4-dimethyl-N-(quinolin-5-ylmethyl)-1,3-thiazol-2-amine
1-(2-cyclopropylphenyl)-3-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]urea
4-(2-methyl-1,3-benzothiazole-5-carbonyl)-1λ6-thiomorpholine-1,1-dione
6-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-N-(propan-2-yl)pyrimidin-4-amine
4-(1H-pyrazol-1-yl)-1-(pyridine-3-sulfonyl)piperidine-4-carboxylic acid
(1R,5R)-3-[4-(piperidin-1-ylmethyl)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-7-chloro-4-methylquinolin-2-amine
N-[(1S,2S)-2-hydroxycyclohexyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
4-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-1λ6-thiomorpholine-1,1-dione
2-methyl-1-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidine
6-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]pyridine-2-carboxylic acid
8-[(5-ethylpyridin-2-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
{[4-(3-chlorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]methyl}(furan-3-ylmethyl)methylamine
(1S,5R)-6-(cyclopropylmethyl)-3-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4S)-4-(4-{[(4-tert-butylphenyl)formamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
2-(4-acetyl-1,4-diazepan-1-yl)-2-(2-fluoro-5-methoxyphenyl)acetic acid
6-methyl-5-[5-(1-methylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
ethyl 4-({4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-1H-pyrazole-3-carboxylate
4-{3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(quinolin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
9-[3-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)propanoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
7-[(3-methylphenyl)methyl]-2-(thian-4-yl)-2,7-diazaspiro[4.5]decan-6-one
cyclopentyl 4-({[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]carbamoyl}amino)benzoate
6-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
1-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-4-(1H-pyrazol-4-yl)butan-1-one
5-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
7-{3-[(pyridin-3-yl)amino]propyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-[4-(ethylcarbamoyl)-2-methylphenyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carboxamide
3-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1-(1-propyl-1H-1,2,3-triazol-4-yl)urea
1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-2-methyl-1,4-diazepan-5-one
(2R,6R)-4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
{4-[(4-chlorophenyl)methyl]-1-(quinoxalin-2-yl)piperidin-4-yl}methanol
7-(5-methylthiophen-2-yl)-4-(morpholine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one