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4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine-1-sulfonamide
1-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-(9H-carbazol-3-yl)ethan-1-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl){[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}amine
3-{5-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-[(5-chlorothiophen-2-yl)methyl]-1-{4-[(dimethylsulfamoyl)amino]phenyl}piperidin-4-amine
6-{1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}pyrimidin-4-ol
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(2-oxopiperidin-1-yl)acetamide
5-[2-(4-fluorophenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-cyclobutanecarbonyl-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]piperidine-4-carboxamide
{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-2,5-dihydro-1H-pyrrole-2-carboxamide
1-(4,6-dimethylpyrimidin-2-yl)-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}piperidin-4-amine
N-methyl-N-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}thian-4-amine
N-(1H-1,2,4-triazol-3-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-(2-fluorobenzoyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
6-fluoro-3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
2-{4-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1-(4-chloro-3-methylbenzoyl)-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
[(5-chloro-2,3-dimethoxyphenyl)methyl]({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
3-(azonan-1-ylmethyl)-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(1,2,4-oxadiazol-3-yl)piperidine
1-[(2E)-2-methylbut-2-en-1-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[(3R,4S)-1-{[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(2R,6R)-10-methoxy-4-propanoyl-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-[(4-fluorophenyl)methyl]-1-[(5-methyl-1,2-oxazol-3-yl)methyl]piperidine
N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
4-amino-N-[(3-chlorophenyl)methyl]-N-(2-methylpropyl)pyridine-2-carboxamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-3-(methylsulfanyl)propanamide
ethyl 2-(2-{[1-(cyclohexylmethyl)-1H-1,2,3-triazol-4-yl]formamido}ethyl)-1,3-thiazole-4-carboxylate
N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(3-phenylphenyl)piperidin-4-amine
7-(thiophen-2-yl)-4-{[4-(trifluoromethoxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2R,6S)-2,6-dimethyl-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}morpholine
4-(2H-1,3-benzodioxol-5-yl)-2-[5-cyclopropyl-4-(4-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-3-(thiophen-3-yl)propanamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-methyl-N-(quinolin-4-ylmethyl)acetamide
1-(oxolan-2-ylmethyl)-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
1-[4-(1H-imidazol-1-yl)phenyl]-3-[1-(morpholin-4-ylmethyl)cyclopentyl]urea
[(3,4-dimethoxyphenyl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
5-(2-chlorophenyl)-2-methyl-N-[3-(pyridin-4-yl)propyl]furan-3-carboxamide
1,7-dimethyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-indole-2-carboxamide
2-[(1-methyl-1H-indol-2-yl)methyl]-9-oxa-2-azaspiro[5.5]undecane
1-{1-[4-(4-fluorophenyl)-4-oxobutanoyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
N-[2-(3-ethylphenoxy)ethyl]-4-hydroxy-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[(4-methylphenyl)sulfanyl]-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperidin-4-yl)methanol
3-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-methyl-3-(pyridin-3-yl)-4-[(1s,4s)-4-aminocyclohexyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one