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N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-butoxyacetamide
4-ethyl-3-[1-(4-methoxy-3,5-dimethylbenzoyl)piperidin-3-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[4-(2-methyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]-1,3-benzothiazole
4-chloro-N-[1-(pyridin-4-yl)propan-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(2-methoxyethyl)-N-[(2-methoxyphenyl)methyl]-5-oxo-N-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
1-(4-aminopyrimidin-2-yl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
6-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-1H-indole
N-[2-(dimethylamino)ethyl]-N-methyl-3-({1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}oxy)benzamide
1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepan-6-ol
4-{3-cyclopropyl-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazole-5-carbonyl}morpholine
(2R,6S)-2,6-dimethyl-4-(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)morpholine
1-(2,5-dimethylphenyl)-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazine
4-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(propylsulfanyl)acetamide
1-[1'-(2,3-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
(1S,5R)-6-(5-chlorothiophene-2-carbonyl)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
1-butyl-3-[2-(methylsulfanyl)ethyl]-5-(1,2-oxazol-3-yl)-1H-1,2,4-triazole
3-(2-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-indole
1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-4-(propan-2-yl)-1,4-diazepane
N-cyclopropyl-1-(3-methylfuran-2-carbonyl)piperazine-2-carboxamide
({2-[(2-chloroprop-2-en-1-yl)oxy]-7-fluoroquinolin-3-yl}methyl)(furan-2-ylmethyl)amine
(4aS,7aR)-N-(2,4-dimethoxyphenyl)-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
ethyl 5-[(3,4-dimethoxyphenyl)methyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-[4-phenyl-5-(2,4,5-trifluorophenyl)-1H-imidazol-1-yl]butan-1-amine
N-(2-methoxyethyl)-4-methyl-3-{[(1H-1,2,4-triazol-3-ylmethyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[3-oxo-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-4-carbonitrile
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-phenylazepane-1-carboxamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-5-methyl-1H-indazole-3-carboxamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-methanesulfonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(1-phenyl-1H-pyrazol-5-yl)urea
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenyl-1,4-diazepane
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(pyridin-2-yl)acetamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(4-hydroxypiperidin-1-yl)ethyl]acetamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methylfuran-3-carbonyl)piperidine
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
3-{[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[2-(dimethylamino)ethyl]-5-(furan-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(2S,4S)-4-amino-N-methyl-1-(2-methyl-1,8-naphthyridine-3-carbonyl)pyrrolidine-2-carboxamide
3-methyl-1-propyl-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-4-carboxamide
(4aS,8aR)-6-(5-fluoropentyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
4-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-6-methoxypyrimidine
N-(1-{1-[3-(furan-2-yl)propanoyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methyl-3-(methylsulfanyl)propanamide
N-[2-(dimethylamino)ethyl]-4-methyl-N-[(3-methylthiophen-2-yl)methyl]-1,3-oxazole-5-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-(4-acetylphenoxymethyl)-N-(butan-2-yl)-N-ethyl-1,2-oxazole-3-carboxamide
3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N'-cycloheptyl-N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]butanediamide
2-amino-N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-6-(propan-2-yl)pyrimidine-4-carboxamide
methyl 5-{[(4-acetamidophenyl)methyl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate