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4-{3-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]propoxy}benzamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(propan-2-yl)benzamide
5-{3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}quinoxaline
5-(4-formyl-1,4-diazepan-1-yl)-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-ethyl-2,3-dimethyl-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-(furan-3-carbonyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-3-(1-methylpiperidin-2-yl)propanamide
1-phenyl-3-[4-(pyrazin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-(2,5-dioxoimidazolidin-1-yl)acetamide
1-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-phenoxypiperidine-4-carboxylic acid
3-(furan-2-yl)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
6-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]pyrimidin-4-amine
(2S,4S)-4-amino-1-(2,3-dihydro-1H-indene-2-carbonyl)-N-methylpyrrolidine-2-carboxamide
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propane-2-sulfonyl)piperidine
(1S,2S,3R,4R)-3-[4-(4-methylphenoxy)piperidine-1-carbonyl]bicyclo[2.2.1]heptan-2-amine
1-phenyl-5-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1H-1,2,3,4-tetrazole
N-cyclopropyl-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[(2-methoxyphenyl)methyl]butanamide
4-methyl-N-(3-{8-oxo-2-oxa-7-azaspiro[4.5]decan-7-yl}propyl)benzene-1-sulfonamide
3-[(3R,4S)-4-(dimethylamino)-1-[(1-methyl-1H-indol-6-yl)methyl]piperidin-3-yl]propan-1-ol
2-amino-3-ethyl-N-{[3-(trifluoromethyl)phenyl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
methyl 4-({[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]carbamoyl}amino)benzoate
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
4-[6-(2-chloro-4-fluorophenyl)pyridine-3-carbonyl]morpholine
N-[(2-cyclohexylpyrimidin-5-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
[(3R,4R)-1-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-(2,6-dimethylpyridin-3-yl)-2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidine
1-{1'-[(3,4-difluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
(4S)-3-[2-(4-benzoylpiperidin-1-yl)-2-oxoethyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
N-(4-methoxyphenyl)-3-(4-phenylbenzoyl)piperidine-1-carboxamide
3-{5-[2-hydroxy-4-(methylsulfanyl)butanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(propan-2-yl)propanamide
5-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
5-[2-(2-methyl-1H-imidazol-1-yl)propanoyl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]pyrazine-2-carboxamide
6-(5-chloro-2-methoxypyridin-4-yl)-N-ethyl-N-methylpyrimidin-4-amine
4-{1-[(2-fluoro-5-methylphenyl)methyl]azetidin-3-yl}pyridine
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-N-(2-ethylphenyl)piperidine-1-carboxamide
N-methyl-2-{1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-4-yl}acetamide
(1S,9aR)-1-{[4-(methoxymethyl)piperidin-1-yl]methyl}-octahydro-1H-quinolizine
(3S,4S)-1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
4-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1-methyl-1H-indole
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3-{2-[1-(1H-indole-6-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-(4-methoxyphenyl)-6,6-dimethyl-4-[2-(methylsulfanyl)acetyl]piperazin-2-one
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-2-[2-(thiophen-2-yl)ethyl]piperidine
3-[6-hydroxy-4-(1H-imidazol-4-ylmethyl)-1,4-diazepane-1-carbonyl]benzonitrile
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
5-{4-[(2-hydroxy-6-methylquinolin-3-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
4-{3-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]piperidin-1-yl}-2-(3-methoxypropyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-4-(1H-pyrrol-1-yl)phenol