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2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(1H-imidazol-4-yl)ethyl]acetamide
N-(2,4-dimethoxyphenyl)-3-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
3-{2-[(2S)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
(1S,5R)-3-{[3-(furan-2-yl)phenyl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
3-[(1S,2S)-2-hydroxycyclohexyl]-1-[4-(3-methoxyphenoxy)phenyl]urea
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
6-methyl-2-propyl-5-[5-(pyridazin-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
5-ethyl-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methylpyrimidin-4-amine
2-[3,5-dimethyl-1-(pyrimidin-5-yl)-1H-pyrazol-4-yl]phenol
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-methylacetamide
N-benzyl-6-(3,4-dimethylpiperazin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(3-phenylpropyl)piperidine
3-[({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1λ6-thiolane-1,1-dione
2-[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-2-yl]ethan-1-ol
1-{3-oxo-3-[4-(quinazolin-4-yl)piperazin-1-yl]propyl}-1,2-dihydropyridin-2-one
1-{[2-(cyclopentyloxy)phenyl]methyl}-4-methoxypiperidine
N-[2-(diethylamino)ethyl]-N-ethyl-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
ethyl 4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-5-methyl-1,3,4-oxadiazol-2-amine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2,6-dimethyl-N-(oxolan-2-ylmethyl)pyrimidine-4-carboxamide
1-benzoyl-4-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperazine
2-(3-fluorophenyl)-N-[(1R,2S)-2-phenylcyclopropyl]-1,3-benzoxazole-5-carboxamide
(4aS,8aR)-6-[4-(trifluoromethyl)pyridin-2-yl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
5-{1-[2-(2-chloro-6-fluorophenyl)-1H-imidazol-1-yl]ethyl}-3-propyl-1,2,4-oxadiazole
5-(5-methylpyridine-3-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(2-propoxybenzoyl)piperidin-4-ol
4-(2-phenylethyl)-1-(quinolin-2-yl)piperidine-4-carboxylic acid
5-[({1-[4-(3-fluorophenyl)phenyl]piperidin-4-yl}amino)methyl]-1-methylpyrrolidin-2-one
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(morpholin-4-yl)-2-oxoethyl]pyrrolidine-3-carboxylic acid
1-[2-hydroxy-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]ethan-1-one
methyl 4-[5-(2-methoxy-2-phenylacetamido)-1H-pyrazol-1-yl]piperidine-1-carboxylate
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-chlorobenzamide
N-[2-(1H-imidazol-4-yl)ethyl]-3-(2-methoxyphenyl)benzamide
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[3-(pyrrolidin-1-yl)propyl]acetamide
N-ethyl-2-(4-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)pyrimidin-4-amine
N-(3-{[(3-hydroxypropyl)[(4-methylphenyl)methyl]carbamoyl]amino}-4-methylphenyl)acetamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-{[(furan-2-ylmethyl)amino]methyl}-3-hydroxypiperidin-2-one
1-(prop-2-en-1-yl)-2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H-imidazole
2-methyl-5-(4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
5-(3-chloro-4-methylbenzoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
N,N-dimethyl-2-{[(6-methyl-2-propylpyrimidin-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-ethyl-1-(1H-pyrazole-4-carbonyl)piperidine-3-carboxamide
[(4aS,8aR)-6-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-4a-yl]methanol
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
1-methanesulfonyl-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-({3-[2-(pyridin-2-yl)-1H-imidazol-1-yl]phenyl}methyl)propanamide
1-[2-(3,4-dimethylphenoxy)ethyl]-3-methoxy-1,2-dihydropyridin-2-one
2-propyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyridine-4-carboxamide
8-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione