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N,5,7-trimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-benzyl-N-ethyl-5-(morpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[2-(dimethylamino)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
1-{3-[2-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
4-{3-[1-(dimethylamino)ethyl]phenyl}-N,N-dimethylbenzamide
5-ethyl-2,3-dimethyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-methyl-3-propyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-pyrazole-5-carboxamide
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-propoxyethan-1-one
N-{2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}aniline
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-benzyl-4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(benzenesulfonyl)-N-(4,4,4-trifluorobutan-2-yl)piperidin-4-amine
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-2-(pyrrolidin-1-yl)-6-(thiophen-3-yl)pyridine-3-carboxamide
7,7-dimethyl-2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-tert-butyl-4-[4-(2-fluoro-4-methoxyphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]acetic acid
N-cyclohexyl-N-(pyridin-4-ylmethyl)-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-cyclopropyl-1-{1-[4-(ethylamino)pyrimidin-2-yl]piperidin-4-yl}piperidine-3-carboxamide
(2S)-3-(pyridin-4-yl)-2-[(3,5,7-trimethyl-1H-indol-2-yl)formamido]propanoic acid
5-[4-(diphenylmethyl)piperazin-1-yl]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(8-methoxyquinolin-2-yl)methyl]-4-phenylpiperidine-4-carbonitrile
1,3-dimethyl-2,6-dioxo-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
[4-(2,4,5-trimethoxybenzoyl)-1,4-oxazepan-6-yl]methanol
3-(2-methoxyethyl)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxylic acid
(2S,4R)-4-amino-N,N-diethyl-1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidine-2-carboxamide
4-{[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}pyridin-2-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-phenoxybenzamide
5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-{1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}benzoic acid
N-{1-[1-(furan-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
1-(3,4-dimethoxyphenyl)-2-{1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethan-1-amine
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}oxan-4-amine
1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-(pyridin-2-yl)-1H-1,3-benzodiazole
[(3R,4R)-4-[(dimethylamino)methyl]-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
3-{1-[(1-cycloheptanecarbonylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-1-ol
2-amino-7-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]pyridine-2-carboxylic acid
5,6-dimethyl-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-oxo-2-(2-phenylindolizin-3-yl)acetamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
1-cyclopropyl-N-methyl-5-oxo-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-3-carboxamide
2-{2-[(2-methyl-3-oxopiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetic acid
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
N-(1-{1-[2-(trifluoromethyl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-methyl-N-[2-(oxolan-3-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(6-methylpyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-cyclohexyl-N-[(4-methoxy-2,5-dimethylphenyl)methyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide