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2-(6-methoxypyridin-3-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]propanamide
3-(1H-1,2,3-benzotriazol-4-yl)-1-[1-(3,4-diethoxyphenyl)ethyl]urea
N-[(4-fluorophenyl)methyl]-3-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)propanamide
(2S)-2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-2-phenylethan-1-ol
N,N-dimethyl-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazine-1-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
methyl 3-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[methyl(2-methylpropyl)amino]methyl}piperidin-2-one
1-(2-phenoxyethyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine
N-({4-[4-(furan-2-carbonyl)piperazin-1-yl]quinazolin-2-yl}methyl)-N-(prop-2-yn-1-yl)cyclohexanamine
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(oxan-4-ylmethyl)pyridin-2-amine
1-[3-(cycloheptylamino)propyl]piperidine-4-carboxamide
N-(1-hydroxybutan-2-yl)-3-(1-methyl-1H-pyrazol-4-yl)-N-[(5-methylthiophen-2-yl)methyl]propanamide
1-[2-(3-chlorophenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-ethyl-N-(2-hydroxyethyl)piperidine-3-carboxamide
N-methyl-2-[3-(methylsulfanyl)phenyl]pyridine-4-carboxamide
3-fluoro-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
4-(methoxymethyl)-6-(2-phenylphenyl)pyrimidine
4-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,6-dimethylpyrimidine
methyl (2S)-1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(morpholin-3-yl)ethan-1-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
4-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-6-fluoro-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}benzamide
2-(2-chloro-6-fluorobenzoyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(propan-2-yloxy)acetamide
5-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[1-(1,3-thiazol-5-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-[3-(trifluoromethoxy)phenyl]-1H-imidazole
8-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
(3S,4R)-4-(4-fluorophenyl)-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidine-3-carboxylic acid
1-(2-ethoxypyridine-3-carbonyl)-4-[(2-fluorophenyl)methyl]-1,4-diazepane
3-{3-ethyl-5-[5-(1H-pyrazol-1-ylmethyl)furan-2-yl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[2-(pyridin-3-yloxy)ethyl]benzamide
2-(2-fluoro-5-methoxyphenyl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
(3R,4R)-1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
ethyl 1-{[4-(4-acetyl-1,4-diazepan-1-yl)-8-methylquinazolin-2-yl]methyl}piperidine-2-carboxylate
N-ethyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-phenylacetamide
N-(1-hydroxy-3-methylbutan-2-yl)-2-methyl-1-benzofuran-5-carboxamide
3-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-5-fluorobenzonitrile
5-methoxy-9-[3-(1H-pyrazol-4-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecane
3-chloro-6-methyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-[1-(4-fluorophenyl)ethyl]-N-methyl-1,2-oxazole-3-carboxamide
(4aS,8aS)-2-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-decahydroisoquinolin-4a-ol
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-ethyl-1-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]urea
N-(2-methylpropyl)-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-(3-phenylprop-2-yn-1-yl)acetamide