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1-[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyrimidin-2-amine
2-[4-(3-chloro-5-fluoro-4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]propanoic acid
5-chloro-2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-{1-[(8-methylquinolin-5-yl)methyl]pyrrolidin-3-yl}acetamide
(2S)-2-[2-(2,4-dimethylbenzenesulfonamido)acetamido]-3-phenylpropanoic acid
1-(2-chlorophenyl)-3-{1-[1-(2-methoxyethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3,7-dimethyl-11-(4,5,6,7-tetrahydro-1,3-benzothiazole-2-carbonyl)-3,7,11-triazaspiro[5.6]dodecane
2-[4-(2-ethoxy-2-oxoethyl)piperazin-1-yl]quinoline-4-carboxylic acid
1-methyl-4-[2-(methylamino)pyridine-4-carbonyl]-3-(propan-2-yl)piperazin-2-one
4-methanesulfonyl-2-(naphthalen-1-ylmethyl)morpholine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(1-methyl-1H-indol-3-yl)acetamide
{[3-(4-fluorophenyl)oxolan-3-yl]methyl}({[6-(trifluoromethyl)pyridin-3-yl]methyl})amine
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[1-(pyrazin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[3-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
methyl 2-(5-methyl-2-{[(5-methylpyrazin-2-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
N'-[(3-chlorophenyl)methyl]-N'-(2-methylpropyl)-N-(1,3,4-thiadiazol-2-yl)ethanediamide
1-methyl-4-{2-methyl-1H-imidazo[4,5-b]pyridin-6-yl}-1H-pyrrolo[2,3-b]pyridine
(3S,9aR)-3-(cyclohexylmethyl)-8-(3-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aR,7aS)-1-(2-methoxyacetyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazin-1-yl)pyrimidine
1-[2-(2,3-dimethoxyphenyl)acetyl]-3-propylpiperidine-3-carboxylic acid
2-(furan-2-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(5-phenylthiophen-2-yl)methyl]pyrrolidin-3-amine
1-(2-methoxy-4-{[(1-methylpiperidin-4-yl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
N-{4-[2-(2-methoxyethyl)morpholine-4-carbonyl]-3-methylphenyl}acetamide
N-(2-hydroxy-3-phenoxypropyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-[1-({2-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)pyrrolidin-2-yl]pyridine
(3aS,6aS)-2-cyclopentyl-5-[4-(methylsulfanyl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[(8-hydroxyquinolin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-ethyl-1-methyl-3-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]propanamide
(2R,3R)-3-(dimethylamino)-1'-[(2,5-dimethylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(3S,9aR)-3-(cyclohexylmethyl)-8-(3,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine-4-carboxylic acid
4-[4-(azetidine-1-carbonyl)phenoxy]-N,N-dimethylpiperidine-1-sulfonamide
5-(diethylamino)-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
N-[4-(2-fluorophenoxy)phenyl]-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxamide
2-(2-aminoethyl)-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinazolin-4-amine
4-ethyl-1-(1-methyl-1H-indole-2-carbonyl)-1,4-diazepan-5-one
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrimidin-2-amine
ethyl 1-[4-(pyridin-3-yl)pyrimidin-2-yl]piperidine-3-carboxylate
2-{[1-(furan-3-ylmethyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
dimethyl({4-methyl-5-[1-(pyridin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
(1S,5R)-6-benzyl-3-(3-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-oxo-3-(pentan-3-yl)-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
[(4-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-oxazepan-6-yl)methyl]dimethylamine