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7-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(1-acetylpiperidin-4-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
N-[(2,5-difluorophenyl)methyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
(4aS,7aR)-1-(benzenesulfonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
2,3-dimethyl-7-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
6-methoxy-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidin-4-amine
[5-({7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)furan-2-yl]methanol
N-[2-(dimethylamino)ethyl]-1-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N1-(4-methylpyridin-2-yl)-N2-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]ethane-1,2-diamine
N-[(4-methoxyphenyl)methyl]-N-propylquinoxaline-6-carboxamide
3-{[1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methyl}benzamide
1-{2-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-(1-cyclopentyl-1H-pyrazol-5-yl)-2-[2-(pyridin-2-yl)ethyl]piperidine-1-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(propylcarbamoyl)piperidine-4-carboxylic acid
2-(2-aminoethyl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}quinazolin-4-amine
(3S,9aR)-8-(2-methoxybenzoyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-[1-(1H-pyrazol-1-yl)propan-2-yl]urea
2-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)acetamido]-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]urea
6-(1-methylpiperidin-3-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-4-amine
3-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}pyridin-2-amine
N-(2-ethoxyphenyl)-2-methyl-4-[(4-methylphenyl)methyl]-3-oxopiperazine-1-carboxamide
3-{4-[3-(5-methylfuran-2-yl)butyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
1-propyl-2-[1-(thiophen-2-ylmethyl)-1H-imidazol-2-yl]-1H-imidazole
2-(4-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1,3-thiazol-2-yl)pyrimidine
8-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
(2S,3R)-3-hydroxy-2-({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}amino)butanamide
1-{4-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidine-1-carbonyl]phenyl}ethan-1-one
1-[(2-butyl-1H-imidazol-4-yl)methyl]-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
N-cyclobutyl-4-{methyl[2-(methylcarbamoyl)ethyl]sulfamoyl}benzamide
(2R,3R,6R)-3-(3-hydroxyphenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
6-tert-butyl-2-oxo-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2,3-dihydropyrimidine-4-carboxamide
{4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]morpholin-3-yl}methanol
2-[2-(dimethylamino)ethyl]-9-(2,4-dimethylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-4-[(2,6-dichloro-3-hydroxyphenyl)methyl]piperazine-2-carboxamide
3-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]-6-(propan-2-yloxy)pyridazine
N-methyl-2-(naphthalen-2-yloxy)-N-(quinoxalin-6-ylmethyl)propanamide
7-methoxy-3-[5-(piperidine-1-carbonyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1H-3-benzazepine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(6-ethylpyrimidin-4-yl)piperidin-3-ol
1-{4-[4-(3,4-dimethylpiperazine-1-carbonyl)-2-methoxyphenoxy]piperidin-1-yl}ethan-1-one
2-amino-4-[2-(morpholin-4-yl)-1,3-thiazol-5-yl]-6-phenylpyridine-3-carbonitrile
(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)methanol
1-(cyclopropylmethyl)-N-methyl-5-(naphthalene-1-carbonyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1H-1,2,3-triazole-5-carboxamide
2-(2-methoxyethoxy)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2,7,8-trimethyl-N-(5-oxo-1-propylpyrrolidin-3-yl)quinoline-4-carboxamide