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N-[(5-chlorothiophen-2-yl)methyl]-1-methylazepane-2-carboxamide
2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-indole
N'-(2,4-dimethoxyphenyl)-N-(2-methylprop-2-en-1-yl)propanediamide
3-chloro-N-(2-methoxyethyl)-4-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}oxy)benzamide
1-(2-aminoethyl)-N-methyl-N-(quinolin-5-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-benzyl-4-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]-1,4-diazepan-6-ol
1-(6-cyanopyridin-3-yl)-3-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]urea
(1S,5R)-6-[(3-fluoro-2-methylphenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-benzyl-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxylic acid
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-thiazole-4-carboxamide
2-methyl-3-({[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]carbamoyl}amino)benzamide
2-({[(3R,4R)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-2-methyl-N-(pyridin-3-ylmethyl)propanamide
3-(2-fluorophenyl)-5-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,4-oxadiazole
4-ethyl-1-methyl-3-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(2-methyloxane-2-carbonyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
1-{3-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-[(5-methylfuran-2-yl)methyl]-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,N-dimethyl-5-(1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-1H-imidazol-2-yl)pyrimidin-2-amine
(4aS,8aR)-6-(1-benzofuran-2-ylmethyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
1,5-dimethyl-4-({2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-(ethylcarbamoyl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-{[(1r,4r)-4-hydroxycyclohexyl]carbamoyl}pyrrolidine-2-carboxylate
2-[(2E)-3-phenylprop-2-en-1-yl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(4-acetylpiperazin-1-yl)-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
N-(cyclobutylmethyl)-7-(2-methoxyacetamido)-1-methyl-N-(oxolan-2-ylmethyl)-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
1-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4-oxo-1,4-dihydroquinoline-3-carboxamide
N-methyl-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-(naphthalen-1-ylmethyl)propanamide
2-{4-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]piperidin-1-yl}acetamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3-[(3-methylbut-2-en-1-yl)amino]-5-[(propan-2-yl)sulfamoyl]benzamide
8-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-oxa-8-azaspiro[4.5]decan-3-ol
ethyl 4-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}-1H-pyrazole-3-carboxylate
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
5-methyl-N-[2-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)propyl]thiophene-2-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-6-methylpyridine
3-{[4-(1-hydroxy-2-methylpropyl)piperidin-1-yl]methyl}-6-methyl-1,2-dihydroquinolin-2-one
3-methyl-1-[1-(6-{[(5-methyl-1H-pyrazol-3-yl)methyl]amino}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-[(1-cyclohexylpyrrolidin-3-yl)methyl]-4-methylpyrimidin-2-amine
N-(2-benzylphenyl)-3-(2-oxopyrrolidin-1-yl)piperidine-1-carboxamide
2-(3,5-dimethyl-4-{3-methyl-1-[(3-methylphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazol-1-yl)ethan-1-ol
1-{4-[3-(3-hydroxypropyl)-4H-1,2,4-triazol-4-yl]phenyl}ethan-1-one
1-({4-methyl-5-[1-(pyridin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
4-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-4-oxobutanamide
4-(naphthalen-2-yloxy)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylic acid
1-methyl-3-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-ethoxy-3-{[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one