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1-(2-{[(4-tert-butyl-1,3-thiazol-2-yl)methyl]amino}pyrimidin-4-yl)piperidin-3-ol
2-methyl-3-(2-{[6-(1-methylpiperidin-4-yl)pyrimidin-4-yl]amino}ethyl)-1H-indole-5-carbonitrile
(4aS,7aR)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-amine
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[(4-methoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
5-[3-(benzyloxy)propyl]-3-(oxolan-3-yl)-1H-1,2,4-triazole
(3S,5R)-N5-(4-fluorophenyl)-N3,N3-dimethyl-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
[4-(4-aminopyridin-2-yl)phenyl]methanol
N-[4-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)thiophene-2-carboxamide
1-{3-oxo-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carbonyl}cyclopropane-1-carboxamide
1-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-2-(2,3-dihydro-1H-inden-1-yl)ethan-1-one
N-[6-methyl-5-(1-{[(1-methyl-1H-indazol-3-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridin-2-yl]propanamide
ethyl 4-[4-(4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-hydroxybutyl)piperidine-4-carboxamide
2-methyl-5-[4-(1-propanoylpiperidine-3-carbonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2H-1,3-benzodioxole-5-carboxamide
1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
4-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butanoic acid
N-[4-({2-[(3-methoxyphenyl)methyl]morpholin-4-yl}methyl)phenyl]acetamide
3-(1H-indol-3-yl)-N-[2-(1H-1,2,4-triazol-1-yl)propyl]propanamide
2-methoxy-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)benzamide
7-[3-(3-methoxyphenoxy)propyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-[(isoquinolin-5-yloxy)methyl]-N-[(1R,2S)-2-phenylcyclohexyl]-1,2-oxazole-3-carboxamide
1-(4-cyanobenzoyl)-4-phenoxypiperidine-4-carboxylic acid
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-[(2-ethoxyphenyl)methyl]-N-ethyl-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]urea
2-chloro-4-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenol
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[3-(propan-2-yloxy)phenyl]-4-(9H-purin-6-yl)piperazine-1-carboxamide
1-methyl-3-(1-propyl-1H-1,2,3-triazol-4-yl)-1-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}urea
8-[(2S)-2-hydroxypropanoyl]-3-{2-[methyl(2-methylpropyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-methoxy-4-methylphenoxymethyl)-N-[(3-methylpyridin-4-yl)methyl]-1,3-oxazole-4-carboxamide
5-[2-(1H-imidazol-1-yl)ethyl]-1-[(2-methylphenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
1-[2-hydroxy-3-(4-methoxy-2-{[(2,2,2-trifluoroethyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
3-phenyl-1-[1-(quinoline-2-carbonyl)piperidin-3-yl]propan-1-one
methyl 4-(methylsulfanyl)-2-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}butanoate
5-fluoro-2-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1-methyl-1H-indole
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
1-(4-chloro-3-methylbenzoyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide
({5-[1-(2,6-dimethoxypyridine-3-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-[(2-hydroxyethyl)({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
(3S,7S)-5-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-triene-3-carboxylic acid
[1-({1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
(3aR,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-[2-(1H-1,2,4-triazol-1-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one