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1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-{[(prop-2-en-1-yl)amino]methyl}-1,2-dihydroquinolin-2-one
3-(2-hydroxyethyl)-5-(3-methylbutyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-cyclopropyl-N-{[2-(2,3-dimethoxyphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-{4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
3-({[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amino}methyl)-N,N-dimethylpyridin-2-amine
ethyl 3-({1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)heptanoate
1-methyl-4-(6-methylpyridazin-3-yl)-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-4-(2-oxopyrrolidin-1-yl)benzamide
N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
N-{1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]azepan-3-yl}-5-hydroxypyrazine-2-carboxamide
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-N-(3,5-dimethoxyphenyl)propanamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
[2-(4-methoxyphenyl)ethyl][(2-methylphenyl)methyl][(1-methylpiperidin-4-yl)methyl]amine
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
5-(2-methoxynaphthalen-1-yl)-1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazole
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamide
1-(pyridin-4-ylmethyl)-4-(thiomorpholine-4-carbonyl)pyrrolidin-2-one
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
2-({[(3R,4R)-1-(2-chloro-4,5-difluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-(2-amino-1,3-thiazol-4-yl)-N-[1-(cyclohex-1-en-1-yl)ethyl]propanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-[2-(methylsulfanyl)propyl]-4-phenyl-1H-imidazole
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-1-phenylmethanesulfonamide
1-[2-hydroxy-5-(quinolin-8-yl)phenyl]ethan-1-one
2-{[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}pyridine-3-carboxylic acid
N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
(1R,3S)-7-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-cyclobutanecarbonyl-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]urea
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
{1-[(3,4-dimethoxypyridin-2-yl)methyl]-3-propylpiperidin-3-yl}methanol
N-methyl-2-phenyl-N-[2-(1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
6-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-2-(pyridin-3-yl)pyrimidin-4-amine
1-(4-cyanonaphthalen-1-yl)-3-{[1-(morpholin-4-yl)cyclopentyl]methyl}urea
3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{3-[(2,4-difluorophenyl)methyl]piperidin-3-yl}methanol
dimethyl({[(3R,4S)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-4-propylpyrrolidin-3-yl]sulfamoyl})amine
9-(2-methyl-1,3-thiazole-4-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{[(4-methoxy-3-methylphenyl)methyl](methyl)amino}ethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
2-[5-(1-methyl-1H-indol-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(2-chlorophenyl)propan-1-one
(2S,4S)-N-ethyl-1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-propanamidopyrrolidine-2-carboxamide
3-[(methylsulfanyl)methyl]-1-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperidine
3-(2,4-dimethylphenyl)-1-(oxan-4-yl)urea
(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanol
4-(4-chlorophenyl)-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]butan-1-one
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid