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1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2H-indazol-2-yl)ethan-1-one
3-[4-(2-methoxyphenyl)piperazin-1-yl]-N-(thiophen-2-ylmethyl)propanamide
N-cyclopentyl-2,5-dimethoxy-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzene-1-sulfonamide
1-benzyl-N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl){[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
6-(3-chloro-2-fluorobenzoyl)-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
4-{4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzoyl}morpholine
(2S,4S)-1-[(2E)-but-2-en-1-yl]-N-ethyl-4-[5-(methoxymethyl)furan-2-amido]pyrrolidine-2-carboxamide
8-{[2-(benzylamino)pyrimidin-5-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(4aS,7aR)-1-(furan-3-carbonyl)-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-hydroxy-N-methyl-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
2-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-(2,3-dihydroxypropyl)-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
2-[1-(2,4-dimethylphenyl)-5-[1-(4-methylpiperazin-1-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-(quinolin-4-ylmethyl)acetamide
8-(2,4-dimethylbenzenesulfonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-(cyclopropylmethyl)-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-{[5-(cyclooctylcarbamoyl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridin-3-yl]formamido}propanoate
N-benzyl-2-(trifluoromethyl)pyrrolidine-1-sulfonamide
5-methyl-2-phenyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-imidazole-4-carboxamide
3-(1,4-diazepan-1-ylmethyl)-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
7-(cyclopropylmethyl)-2-[2-(6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
6-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)pyridine-2-carboxylic acid
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]propan-1-one
N-methyl-5-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
2-{1-[(3-fluoropyridin-4-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
ethyl 1-{1-[2-(3-chloro-4-fluorophenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carbonyl}piperidine-3-carboxylate
(4aS,8aR)-1-(2-aminoethyl)-6-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(furan-2-ylmethyl)-5-methoxybenzamide
2-(2-chlorophenyl)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
8-(5-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]propanamide
methyl 3-(2-chlorobenzamido)-5-{[(2E)-3-(1H-imidazol-4-yl)prop-2-enamido]methyl}benzoate
5-(2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,7S)-N,N-dimethyl-4-oxo-3-[2-(piperidin-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-cyclopropyl-5-(2-methoxynaphthalen-1-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)piperidin-2-one
N-(2-methylphenyl)-3-{[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
5-cyclopropyl-N-ethyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-(2-methylprop-2-en-1-yl)-1H-pyrazole-4-carboxamide
1-(3-fluorobenzoyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
4-[2-(2,5-difluorophenyl)acetyl]-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-{2-[4-(azetidin-1-ylmethyl)phenoxy]ethyl}-3-methylpiperidine
N-[1-(benzenesulfonyl)piperidin-4-yl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[(3S,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
3-{4-[5-(acetamidomethyl)pyridin-2-yl]phenyl}propanoic acid
6-methoxy-2-{2-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,3-benzodiazole