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N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
3-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
ethyl 5-{[4-(4-acetylphenyl)piperazin-1-yl]methyl}-1-(2-chlorophenyl)-1H-pyrazole-4-carboxylate
N-[(3S,4R)-1-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
(1S,5R)-6-(naphthalene-1-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-(methoxymethyl)-5-methyl-3-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1,2-oxazole
4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1-[(2S)-oxolan-2-ylmethyl]-1H-1,2,3-triazole
2-{3-[2-(3-acetylphenyl)pyridin-4-yl]pyrrolidin-1-yl}acetic acid
1-(3-chlorophenyl)-3-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)urea
(1R,5R)-6-benzyl-3-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-(dimethylamino)-N-[2-methyl-5-({[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]carbamoyl}amino)phenyl]acetamide
[(3R,4S)-1-[(4-ethylphenyl)methyl]-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-methyl-4-(6-methyl-2-propylpyrimidin-4-yl)piperazine-2-carboxylic acid
3-(3-{furo[3,2-c]pyridin-4-yl}phenyl)-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazole
N-[(3R,4S)-4-cyclopropyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
N-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-N-(pyridin-3-ylmethyl)cycloheptanamine
N-[(2-fluorophenyl)methyl]-3-[1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]propanamide
2-[2-(methylsulfanyl)phenyl]pyridine-4-carboxamide
N'1-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclopropane-1,1-dicarboxamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-3-(1-methylpiperidin-2-yl)propan-1-one
2-[4-fluoro-3-(hydroxymethyl)phenyl]-2-[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]acetic acid
7-fluoro-3-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}[(2-methoxyphenyl)methyl]methylamine
[4-(2-phenylethyl)-1-(quinolin-2-ylmethyl)piperidin-4-yl]methanol
(3aS,7aR)-5-methyl-2-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-pyrrole-2-carboxamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(3-methoxyphenyl)methyl]-N-methyl-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[(3S,4R)-1-(2,4-dimethylquinoline-7-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
[(1-cyclohexylpiperidin-3-yl)methyl][(4-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
N-[1-(1H-imidazol-2-yl)ethyl]-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N,3-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
1-(5,6-dimethylpyrimidin-4-yl)-N,N-diethylpyrrolidin-3-amine
N-[2-(piperidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
2-[2-(dimethylamino)ethyl]-8-(2-methyl-5-propylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-5-phenyl-N-[1-(pyrazin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
2-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
4-[(2-methylprop-2-en-1-yl)oxy]-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
N-[4-(furan-2-yl)phenyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
4-[3-(morpholin-4-ylmethyl)phenyl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
5-oxo-1-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]pyrrolidine-3-carboxylic acid
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-4-phenylazepane
2-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]benzonitrile
dimethyl({3-[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]propyl})amine
4-{5-[3-(3-methylbutanoyl)piperidine-1-carbonyl]pyridin-2-yl}piperazin-2-one
1-{4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]phenyl}-3,5-dimethyl-1H-pyrazole
N-butyl-3-{imidazo[1,2-a]pyridin-2-yl}-N-(thiophen-3-ylmethyl)propanamide