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(1R,5R)-N-(4-ethoxyphenyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-(2,2-dimethyloxane-4-carbonyl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-methyl-4-({5-[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
(3S,9aR)-8-benzyl-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[6-hydroxy-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-1-yl]-1,3-thiazole-4-carboxamide
3-methyl-4-[5-(oxolan-3-yl)-3-phenyl-1H-1,2,4-triazol-1-yl]pyridine
1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
5-(2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2-ethylbutyl)-8-[2-(3-methylpiperidin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-methyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,3-oxazole-5-carboxamide
4-({1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-2-yl}methyl)morpholine
(2S,4R)-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-hydroxy-N-methylpyrrolidine-2-carboxamide
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-[(2S)-5-oxopyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-benzyl-3-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]benzamide
4,6-dimethyl-3-{3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
(2S)-1-(4-cyano-1-methyl-1H-pyrrole-2-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-[(2-fluorophenyl)methyl]-6-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
8-(3-methyl-1,2-oxazole-5-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-pentanoyl-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
6-[(3-methoxyphenyl)methoxy]-4-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperazine
1-({4-methyl-5-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
ethyl 5-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-methyl-6-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}pyridine-2-carboxamide
2-{[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethan-1-ol
1-(pyrimidin-2-yl)-N-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-amine
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N-(prop-2-en-1-yl)-4-{[2-(pyrrolidin-1-yl)ethyl]sulfamoyl}benzamide
1-[1-({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)piperidin-3-yl]ethan-1-one
6-(2-cyclopentyl-2-phenylacetyl)-N-(furan-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
5-(morpholin-4-yl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-(1-ethyl-8-{[3-(2-methylphenyl)phenyl]methyl}-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl)acetamide
2-amino-6-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyrimidine-4-carboxamide
1-{3-[2-(3-hydroxypropyl)-1H-1,3-benzodiazol-1-yl]phenyl}ethan-1-one
2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-4-methoxybenzoic acid
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-3-(trifluoromethyl)benzamide
1-(1H-indazol-6-yl)-3-[2-(2-methylpropanesulfonyl)ethyl]urea
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylpyrazolo[1,5-a]pyridine-7-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[2-chloro-5-(morpholin-4-yl)phenyl]thiomorpholine-4-carboxamide
[(3-methyl-1H-indol-2-yl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
3-(hydroxymethyl)-1-[(4-methylnaphthalen-1-yl)methyl]piperidin-3-ol
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(4aS,7aR)-1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,N-dimethyl-4-[3-(propan-2-yloxy)phenyl]benzamide