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3-[3-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-1H-indole
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-phenoxyethan-1-one
2-methyl-6-[1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-yl]pyrimidin-4-ol
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
8-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}quinoline
5-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)thiophene-2-sulfonamide
4-(1H-indol-4-yl)-6-(morpholin-4-yl)pyrimidin-2-amine
methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})[2-(1H-pyrazol-4-yl)ethyl]amine
2-(4-chlorophenyl)-4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]morpholine
2-(2,3-dimethylbenzamido)-N-[(1-methylpiperidin-2-yl)methyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
2-{[4-(5-ethylpyrimidin-2-yl)piperazin-1-yl]methyl}-5-fluorophenol
4-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl]benzonitrile
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-6-methylpyridine-2-carboxamide
4-(4-methoxyphenyl)-2-methyl-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
2-{3-[(7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenoxy}ethan-1-ol
(3R,5S)-N-[2-(benzyloxy)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-(2-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethyl)pyridine
(3S,4S)-4-[4-(pyridin-2-yl)piperazin-1-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-ol
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
ethyl 1-[(5-methylthiophen-2-yl)sulfonyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
(1S,5R)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(2-hydroxyethyl)amino)-1λ6-thiolane-1,1-dione
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(5-methylpyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methoxyethyl)-N-methyl-3-[(1-methyl-6-oxopiperidin-3-yl)sulfamoyl]benzamide
2-(2-{1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
(1R,2S)-N-butyl-2-[4-(pyridin-4-yl)piperazine-1-carbonyl]cyclohexane-1-carboxamide
3-{4-[1-(N-methyl-1-thiophen-2-ylformamido)-2-phenylethyl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
2-(2-methylpiperidin-1-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
3-(methoxymethyl)-1-[(2-propoxyphenyl)methyl]pyrrolidine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-[(propylamino)methyl]piperidin-2-one
2-(3-acetyl-1H-pyrazol-1-yl)-N-(1-cyclohexyl-1H-pyrazol-5-yl)acetamide
4-{3-[(phenylsulfanyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}morpholine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2,1-benzoxazole-3-carboxamide
7-(propan-2-yl)-2-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
2-(dimethylamino)-8-[(4-methanesulfonylphenyl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-methyl-4-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,3-oxazole
1-({1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-(pyrrolidin-3-yl)benzamide
2-(2H-1,3-benzodioxol-5-yl)-5-[(2,5-dimethoxyphenyl)methyl]-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
propan-2-yl (3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carboxylate
(3S,4S)-1-{furo[3,2-c]pyridin-4-yl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
4-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-1-(3-chlorophenyl)piperazin-2-one
(2R,6R)-4-[2-(benzenesulfonyl)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-{3-[(4-methoxyphenyl)methyl]-5-{[4-(propan-2-yl)morpholin-2-yl]methyl}-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-methyl-5-({3-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)-1,3-benzothiazole
1-cyclopentyl-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepane