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N-[2-(dimethylamino)ethyl]-2-methyl-7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
3-(azepan-1-ylmethyl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)benzamide
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
1-(3,5-difluorophenyl)-N-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methylpentanamide
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}pyrrolidine-1-carboxamide
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-[(6-methylpyridin-2-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}-4H-chromen-4-one
methyl 2-[3-(2-chlorophenyl)-3-phenylpropanamido]acetate
2-(2-methoxyethyl)-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(1R,9aR)-1-[({[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
N-({5-[(3-chloro-4,5-dimethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
{1-[(3-chloro-4,5-dimethoxyphenyl)methyl]pyrrolidin-3-yl}methanamine
6-[(3aS,6aS)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-octahydropyrrolo[2,3-c]pyrrol-5-yl]-9H-purine
3-cyclopropyl-5-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
2-cyclobutyl-5-(2-methoxyacetamido)-1-methyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
1-{4-[(2-hydroxy-3-methoxypropyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
[(3R,4R)-1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-2-(2-oxopiperidin-1-yl)acetamide
2-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-butyl-1-methyl-4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazin-2-one
2-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-4-carboxamide
1-ethyl-5-methyl-N,N-bis(1,3-oxazol-4-ylmethyl)-1H-pyrazole-4-carboxamide
N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]quinoxaline-6-carboxamide
4-[({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]benzene-1-sulfonamide
3-{[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]amino}butan-1-ol
4-(2H-1,3-benzodioxol-5-yl)-2-[(4-benzylpiperidin-1-yl)methyl]phenol
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
{1-ethyl-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl}(phenyl)methanol
5-methyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-1,3-oxazole-4-carboxamide
N-[5-(thiophen-2-yl)pyridin-2-yl]methanesulfonamide
N-{1-[1-(2-acetamidoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
N-(propan-2-yl)-4-(4H-1,2,4-triazol-4-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-4-(2-phenylethyl)piperidine
5-(2-{2-benzyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)imidazolidine-2,4-dione
1-(4-ethoxyphenyl)-2-{[5-(methoxymethyl)furan-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
(1R,9S)-5-amino-3-[3-(trifluoromethyl)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
1-methyl-3-[(2-oxoazepan-1-yl)methyl]-1,2-dihydroquinolin-2-one
3-methyl-8-[3-methyl-2-(2-methylphenoxy)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-4-(3-methylpyridin-2-yl)piperazine
2,3-dimethyl-7-{[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-[(4-chlorophenyl)sulfanyl]acetamide
1-[3-(cyclopentyloxy)phenyl]-3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]urea
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-ol
({2,5-dimethyl-3-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)[(1-ethyl-1H-pyrazol-4-yl)methyl]methylamine
N-[(8-methoxyquinolin-5-yl)methyl]-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(4aR,7aS)-1-benzyl-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-1-[(3,5-dichloro-2-methoxyphenyl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-[(2-fluorophenyl)methyl]-3-{1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-3-yl}propanamide