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N,N-dimethyl-4-oxo-4-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butanamide
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(3-fluorophenyl)piperidine
2-(1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-thiazole
1'-(1H-1,3-benzodiazole-2-carbonyl)-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-chloro-4-{[1-(3-hydroxypropanoyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
2,2-dimethylpropyl 3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxylate
N-methyl-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-N-(pyrazin-2-ylmethyl)pyridin-2-amine
3-ethyl-N-methyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
1-ethyl-4-[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]piperazin-2-one
N-cyclohexyl-4-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}piperidine-1-carboxamide
(3S)-3-amino-4-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-oxobutanoic acid
4-({1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperidin-4-yl}methyl)morpholine
8-(3-acetylbenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-fluoro-N-(2-{4-oxo-3H,4H-pyrido[3,2-d]pyrimidin-3-yl}ethyl)benzamide
3-[2-(dimethylamino)ethyl]-8-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)-2,2-dimethylpropan-1-ol
N-[2-(morpholin-4-yl)ethyl]-4-(4-{[2-(pyridin-4-yl)ethyl]amino}piperidin-1-yl)benzamide
5-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazine-1-carbonyl)-1H-1,2,3-benzotriazole
1-({3-[(dimethylamino)methyl]phenyl}methyl)-1-methyl-3-(1,3,4-thiadiazol-2-yl)urea
N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
ethyl 3-(2-phenoxyethyl)-1-(1-propylpiperidin-4-yl)piperidine-3-carboxylate
3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-(furan-2-yl)-5-{1-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazol-4-yl}pyrimidine
4-(3-aminopyrrolidine-1-carbonyl)-N-(furan-3-ylmethyl)-N-methylbenzene-1-sulfonamide
5-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrrolidin-2-one
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-4-methyl-1,3-thiazole-5-carboxamide
(2R)-2-amino-3-methoxy-1-[4-(3-methylphenoxy)piperidin-1-yl]propan-1-one
1-ethyl-4-[4-(2-methylpyridin-4-yl)piperazine-1-carbonyl]pyrrolidin-2-one
(2S,4R)-4-{2-[4-(dimethylamino)phenyl]acetamido}-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
1-[(3-fluoro-2-methylphenyl)methyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(2S)-2-(methoxymethyl)-N-[3-(methylsulfanyl)phenyl]pyrrolidine-1-carboxamide
3-methyl-8-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3-hydroxypropyl)-3-[(2-methoxyphenyl)methyl]-1-[2-(methylsulfanyl)phenyl]urea
4-{2-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazole-4-carbonyl}-1,4-oxazepan-6-ol
(2S,5R)-2,5-dimethyl-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
7-(1,3-benzothiazol-2-yl)-4-[1-(4-methoxyphenyl)propan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
1-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carbonyl]-2,3,4,9-tetrahydro-1H-carbazole
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[6-(dimethylamino)pyridin-3-yl]methyl}piperazin-2-one
N-[(1S,2R)-2-aminocyclobutyl]-2-[N-(4-methylphenyl)methanesulfonamido]acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-(2,4-dimethoxyphenyl)-1,2,4-triazin-3-amine
5-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
3-(3,4-dimethoxybenzoyl)-1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
4-phenyl-N-{1-[1-(2-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
2-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)-6-methylphenol
3-(4-benzoyl-6-hydroxy-1,4-diazepan-1-yl)pyrazine-2-carbonitrile
(5S,9aS,9bS)-2-(2-methoxyphenyl)-5-[5-(propan-2-yl)-1H-pyrazol-3-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one