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N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(2-hydroxyphenyl)-N-methylacetamide
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-4-(1H-pyrazol-3-yl)-N-(pyridin-3-ylmethyl)benzamide
5-(3-methoxyphenoxymethyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-3-carboxamide
1-(benzenesulfonyl)-4-(5-phenyl-1,2,4-oxadiazol-3-yl)piperazine
3-(5-chloro-2-methoxybenzoyl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine
4-[4-phenyl-1-(prop-2-en-1-yl)-1H-imidazol-5-yl]pyridine
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrimidin-2-amine
N-[(3S,4R)-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
4-[(2S)-1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]pyrrolidine-2-carbonyl]morpholine
3-[2-(3-chloro-4-hydroxyphenyl)-1H-imidazol-1-yl]-N-(2-methoxyphenyl)propanamide
N-(2-methoxyethyl)-2-methyl-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-1,3-thiazole-4-carboxamide
N-methyl-5-{[6-methyl-2-oxo-4-(trifluoromethyl)-1,2-dihydropyridin-1-yl]methyl}furan-2-carboxamide
7-(2H-1,3-benzodioxol-5-ylmethyl)-2-oxa-7-azaspiro[4.5]decane
(4aS,8aR)-6-[3-(4-methoxyphenyl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
N-[(5-fluoro-2-methylphenyl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
3-(2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
1-{7-[cyclohexyl(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(morpholin-4-yl)propan-1-one
5-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}thiophene-2-sulfonamide
3-({1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}methyl)benzoic acid
4-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}sulfonyl)-N-methylthiophene-2-carboxamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-[2-(methylsulfanyl)acetyl]piperidine-4-carboxylate
N,1-dimethyl-N-[(1-methylpyrrolidin-2-yl)methyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4R)-4-(4-fluorophenyl)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]pyrrolidine-3-carboxylic acid
7-ethyl-2-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
N,N-dimethyl-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-amine
5-acetyl-N-[2-(N-methylmethanesulfonamido)ethyl]thiophene-3-carboxamide
2-{4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(1-methyl-1H-pyrazol-5-yl)acetamide
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(oxane-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,2S,4R)-4-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-ol
4-(3-chloro-4-fluorobenzoyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-(1-benzofuran-5-carbonyl)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
N-[2-(benzyloxy)ethyl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
3-[2-(4-fluorophenyl)ethyl]-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidine
4-{1-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
N-(5-methyl-2-pentanamidophenyl)cyclohex-3-ene-1-carboxamide
2-ethyl-6-[5-(oxolan-2-yl)thiophene-2-carbonyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
4-(2-methoxypyridin-3-yl)-6-(1H-pyrazol-1-yl)pyrimidine
6-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3,4,7-trimethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-indole-2-carboxamide
N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[2-(oxan-4-yl)ethyl]benzamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N,3-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-methyl-1-(oxolan-2-ylmethyl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(4-methyl-1,3-thiazol-2-yl)-4-(6-methyl-9H-purin-9-yl)benzamide
4-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-fluoro-5-sulfamoylbenzamide
(4aS,7aR)-1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
N-benzyl-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide