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N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-4-propylpyrimidine
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-(methylsulfanyl)-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}acetamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-[4-(1H-imidazol-1-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
4-[3-(3-methoxypropyl)piperidine-1-carbonyl]-2-methylphenol
3-benzyl-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1H-1,2,4-triazole
2-({[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}acetamide
1-[2-(1-{3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl)ethyl]-1H-1,2,3,4-tetrazole
1,9-dimethyl-4-(5-phenoxyfuran-2-carbonyl)-1,4,9-triazaspiro[5.5]undecane
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]-N-(cyclohexylmethyl)propanamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
1,5-dimethyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-3-(pyridin-2-yl)propanamide
2-methyl-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-1-benzofuran-5-carboxamide
(2S,3R)-2-amino-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-hydroxybutanamide
3-(4-chloro-2-methylbenzoyl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
{3-[(3-chlorophenyl)methyl]-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methanol
N-(1-benzylpyrrolidin-3-yl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]morpholin-3-yl}acetic acid
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N-(5-methyl-1,2-oxazol-3-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2,3,5,6-tetramethyl-N-[1-(pyridin-4-yl)propan-2-yl]benzamide
2-{3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]piperidin-1-yl}acetamide
2-{4-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
8-(4-chlorobenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(4-ethylpiperazin-1-yl)-N-[2-(1H-imidazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
2-{1-[(3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[1-(pyrimidin-4-yl)ethyl]acetamide
N,N-dimethyl-5-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)pyridin-2-amine
(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)(furan-2-ylmethyl)(prop-2-en-1-yl)amine
5-{[4-(2-methoxybenzoyl)piperazin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methylpyridin-2-amine
ethyl 5-(5-acetylthiophene-2-carbonyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-{1-[1-(5-chloro-2-methoxybenzoyl)piperidin-4-yl]ethyl}morpholine
1-[2-(3-chlorophenyl)ethyl]-4-[(pyridin-2-ylmethyl)amino]pyrrolidin-2-one
4-methyl-N-[3-(methylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-(propan-2-yl)pyrimidine-5-carboxamide
3-(1-ethyl-1H-imidazol-2-yl)-N-(4-methylphenyl)piperidine-1-carboxamide
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-3-(5-amino-1H-1,2,4-triazol-3-yl)propan-1-one
3-cyclopropyl-5-[(2S)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
(3aR,6aR)-2-[(4-chloro-3-fluorophenyl)methyl]-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(1H-indazol-7-yl)-1-{1-oxaspiro[4.4]nonan-3-yl}urea
N-butyl-1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-methylpiperidine-3-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
1-(3-{[2-(dimethylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}propyl)-6-methyl-1,2-dihydropyridin-2-one
6-chloro-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}pyridazin-3-amine
(2E)-3-(3,4-dimethoxyphenyl)-N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]prop-2-enamide
N-(2,5-dimethylphenyl)-3-[3-(trifluoromethyl)benzoyl]piperidine-1-carboxamide
6-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carbonyl}-1,3-benzothiazole