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2-[(1-benzyl-4-phenylpiperidin-4-yl)formamido]acetamide
(1R,5R)-6-(cyclopropylmethyl)-3-(naphthalene-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1-{1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-1H-1,2,3-benzotriazole-5-carboxamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-(2-{[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]amino}propyl)-3,4-dihydroquinazolin-4-one
7-(2-oxopyrrolidin-1-yl)-4-(1-phenyl-1H-pyrazol-5-yl)-1,2,3,4-tetrahydroquinolin-2-one
N-(1-benzothiophen-5-ylmethyl)-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
(2E)-N-{2-[2-(propan-2-yloxy)phenyl]phenyl}but-2-enamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-N-(3-phenylprop-2-yn-1-yl)cyclopropanamine
N-({6-[3-(1-methoxyethyl)phenyl]pyridin-3-yl}methyl)acetamide
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-{2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
1-[2-(piperazin-1-yl)ethyl]-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-amino-4-(3,4-dihydroxyphenyl)-6-(1-propyl-1H-1,2,3-benzotriazol-5-yl)pyridine-3-carbonitrile
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
methyl 3-[(3-{[(4-fluorophenyl)methyl]carbamoyl}-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-yl)amino]propanoate
N-{[1-(6-oxo-1,6-dihydropyridine-2-carbonyl)piperidin-3-yl]methyl}-3-phenylpropanamide
(3S,4R)-1-(4,6-dimethoxypyrimidin-2-yl)-4-(hydroxymethyl)piperidin-3-ol
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-(thiolan-3-yl)urea
1-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
2-chloro-5-acetamido-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]benzamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide
5-{3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
3,5-dimethyl-4-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidin-2-yl}-1,2-oxazole
N-[(5-{[3-(2-aminoethyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
1-benzyl-3-[3-(pyridin-3-yl)propyl]-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-imidazol-2-one
(2S,4S)-4-amino-1-(5-methyl-4-phenylthiophene-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-cyclopentyl-5-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]piperidin-2-one
ethyl 1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(2-phenylethyl)piperidine-4-carboxylate
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
propan-2-yl 2-chloro-5-[(2-methyl-5-oxo-1,4-diazepane-1-carbonyl)amino]benzoate
1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-3-(methylsulfanyl)propan-1-one
8-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)morpholine-4-carboxamide
3-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
1-[3-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyridin-2-yl]piperidin-3-ol
1-(2H-1,3-benzodioxol-5-yl)-5-(dimethyl-1,3-oxazol-5-yl)-3-methyl-1H-1,2,4-triazole
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)pyrrolidin-3-yl]methanol
1-ethyl-4-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}piperazine-2,3-dione
4-[(4-fluorophenyl)methyl]-1-(3-hydroxypropyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(3R,4S)-1-(cyclobutylmethyl)-4-propylpyrrolidin-3-yl]-2-(1H-imidazol-1-yl)acetamide
(1S,3R)-3-amino-N-(2-hydroxyethyl)-N-[(3-methylthiophen-2-yl)methyl]cyclopentane-1-carboxamide
7-fluoro-3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1-(pyridin-4-ylmethyl)-1,2-dihydroquinolin-2-one
5-(2,6-difluorophenoxymethyl)-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide