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2-(4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
5-{3-[1-(cyclobutylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
N-ethyl-5-[1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[(4-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2,2-dimethyloxan-4-yl)-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
1-benzyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}azepan-2-one
2-[1-(2-methyl-1-benzofuran-5-carbonyl)piperidine-3-carbonyl]pyridine
(3R,4R)-4-ethyl-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidine-3,4-diol
(1-methyl-5-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
N-[2-hydroxy-1-(thian-4-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-methyl-N-[2-(oxan-2-yl)ethyl]-2-oxo-4-phenylbutanamide
N-(5-carbamoyl-2-methylphenyl)-4-(1,1-dioxo-1λ6-thiolan-3-yl)piperazine-1-carboxamide
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-1,2-oxazolidin-4-ol
8-(2,5-dimethylbenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-methyl-2-(2-oxo-1,2-dihydropyridin-1-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
2-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)pyridine
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
4-(2-{4-[3-(1H-pyrazol-4-yl)benzoyl]piperazin-1-yl}ethyl)morpholine
1-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
1-(4-methyl-1,3-oxazole-5-carbonyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
2-({[(3R,4R)-1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
5-butyl-1'-(3-methoxypyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cyclooctyl-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]pyrimidin-4-amine
N-[4-(furan-2-yl)phenyl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidine-3-carboxamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(2-methoxyethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
1-[(2-ethylpyrimidin-4-yl)methyl]-4-(2-methylphenyl)-1,4-diazepane
1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
1-(4-fluorophenyl)-4-(4-methoxy-3-methylbenzoyl)-1,4-diazepane
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
6-hydroxy-N-(2-methylquinolin-8-yl)-1,4-oxazepane-4-carboxamide
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-4,6-dimethylpyrimidin-2-amine
(2S,4R)-N-methyl-4-{4-[(2-phenylacetamido)methyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(quinoxalin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,9aR)-1-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
(3aR,6aS)-N-{4-[(2-phenylethyl)carbamoyl]phenyl}-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
1,5,6-trimethyl-3-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-1,2-dihydropyridin-2-one
3-[(3R,4S)-1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(3R,4R)-4-(azepan-1-yl)-1-[(2-methoxyquinolin-3-yl)methyl]piperidin-3-ol
1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-3-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
2-[1-(pyridine-2-carbonyl)azetidin-3-yl]-1H-1,3-benzodiazole
2-[4-(5-ethyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]-1,3-benzothiazole
1-[1'-(5-ethylthiophene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-(pyridin-4-yl)acetamide
3-(2-phenoxyethyl)-8-(pyridine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one