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1-[2-(4-methoxyphenyl)ethyl]-5-(1-methyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-[2-(3-methoxyphenoxy)ethyl]-2-(trifluoromethyl)pyridine
methyl 7-oxo-9-(3-phenylpropoxy)-3-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-benzyl-8-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decan-3-one
1-{2-[({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
N-(6-fluoropyridin-3-yl)-6-hydroxy-1,4-oxazepane-4-carboxamide
(3aR,6aS)-1-oxo-5-[(2-phenylethyl)carbamoyl]-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-ethyl-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1H-pyrazole-4-carboxamide
ethyl 1-[1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]piperidine-4-carboxylate
6,7-dimethoxy-2-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
6-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pent-4-en-1-one
2-methoxy-5-[(4-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperazin-1-yl)methyl]pyrimidine
3-({[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]carbamoyl}methyl)-1,2,3-oxadiazol-3-ium-5-olate
{2-[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]phenyl}methanol
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(9H-purin-6-yl)piperazin-2-yl}ethan-1-ol
2-amino-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)pyridine-4-carboxamide
N-{[1-(2,1,3-benzoxadiazol-4-ylmethyl)pyrrolidin-3-yl]methyl}but-3-enamide
(4aR,7aS)-4-(4-hydroxy-3-methylbenzoyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-{[(2-amino-9H-purin-6-yl)(methyl)amino]methyl}-3,4-dihydroquinazolin-4-one
1-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}piperidin-4-ol
2-(3-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}propyl)phenol
5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-3-(2-phenylethyl)-1H-1,2,4-triazole
2-amino-6-(1-methyl-1H-pyrrol-3-yl)-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
3-{1-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
5-(3-fluorobenzoyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-ethyl-1-{2-[(4-methoxyphenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-N-(prop-2-en-1-yl)cyclopentanamine
(2S,4R)-4-amino-N-methyl-1-{[5-(1,3-oxazol-5-yl)thiophen-2-yl]sulfonyl}pyrrolidine-2-carboxamide
3-[(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)amino]-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
(3aS,6aS)-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2-chloro-4-methoxyphenoxymethyl)-N-ethyl-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-(2-hydroxyethyl)-4-{[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]amino}pyridine-2-carboxamide
(1R,5S,6S)-6-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-oxoacetamide
4-ethyl-3-({1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxylate
2-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-N-(1-methyl-1H-pyrazol-4-yl)acetamide
1-[(1S,5R)-6-{3-[(dimethylamino)methyl]benzoyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
{4-[(2-chlorophenyl)methyl]-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methanol
2-[methyl(pyridin-4-ylmethyl)amino]-1-[4-(3-methylphenoxy)piperidin-1-yl]ethan-1-one
2-[(1-ethylpyrrolidin-2-yl)methyl]-1,2-dihydrophthalazin-1-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]acetamide
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-[(cyclopropylmethyl)sulfanyl]ethan-1-one
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-2,5-dihydro-1H-pyrrole
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-6-methylpyridine-3-carboxamide
2-(4-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide