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N-[1-(4-fluorophenyl)ethyl]-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)ethan-1-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
5-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
4-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-9-(2-hydroxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methylcyclopropanecarbonyl)piperidine
4-(4-chlorophenyl)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-ol
benzyl (7S,9aR)-7-(hydroxymethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
2-(2-ethoxyphenyl)-2-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}acetic acid
5-cyclopropanecarbonyl-1'-(5-ethyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(2,6-dichloro-3-hydroxyphenyl)methyl]-1,4-oxazepan-6-ol
1-[2-(2,2-diphenylethyl)morpholine-4-carbonyl]cyclopropane-1-carboxamide
4-{[(1R,5R)-3-(dimethylsulfamoyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amine
7-(5,8-dimethoxy-4-methylquinolin-2-yl)-4-(furan-2-ylmethyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(methylsulfanyl)propyl]piperidin-3-ol
N-(1-{[(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)piperidin-4-yl]pyridine
2-methyl-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
4-[(1-methyl-1H-imidazol-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1,3,4-oxadiazol-2-amine
3-{4-phenyl-5-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-1H-imidazol-1-yl}propan-1-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(methylamino)pyridine-3-carbonyl]piperidin-3-ol
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
3-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-1-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea
3-(benzyloxy)-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}azetidine
(3S,4S)-4-cyclopropyl-1-[1-(3-methoxyphenyl)piperidin-4-yl]pyrrolidine-3-carboxylic acid
methyl 5-{[(2E)-2-methylbut-2-en-1-yl]amino}-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-{[4-(propan-2-yl)phenyl]methyl}-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
[1-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-3-yl)piperidin-4-yl]methanol
N'-(3-chloro-4-fluorophenyl)-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}propanediamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(1-phenylbutyl)propanamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-(2-methoxyethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
[(3R,4R)-1-[1-(2-chlorophenyl)piperidin-4-yl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[4-chloro-2-(trifluoromethyl)phenyl]-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
N-[(2-chlorophenyl)methyl]-3-[1-(4-methoxybenzoyl)piperidin-3-yl]propanamide
1-{7-[(3E)-pent-3-enoyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine-3-carboxamide
N-[2-(5-methylthiophen-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-4-(1,3-thiazol-2-yl)piperazine
3-(2-ethyl-1H-1,3-benzodiazol-6-yl)-1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}urea
1-methyl-4-[4-(1H-pyrazol-4-yl)butanoyl]piperazine-2-carboxylic acid
4-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperazine-1-carbaldehyde
2-(1-benzofuran-2-yl)-2-[4-(morpholine-4-carbonyl)piperidin-1-yl]acetic acid
2-(3-hydroxyphenyl)-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]acetamide
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-[4-(trifluoromethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{[4-(propan-2-yl)phenyl]methyl}-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)butan-2-ol