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4-(4-methyl-1H-pyrazol-1-yl)-1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidine-4-carboxylic acid
4-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}pyridine
(4aR,8aS)-6-(2-phenylethyl)-1-[2-(1H-pyrazol-1-yl)benzoyl]-decahydro-1,6-naphthyridine
2-(4-fluorophenyl)-2-hydroxy-1-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethan-1-one
5-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-3-(3-methoxyphenyl)-1,2,4-oxadiazole
6-(benzyloxy)-1-(2-methylpropyl)-4-(2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetyl)-1,4-diazepan-2-one
3-(2,4-dimethoxybenzoyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
1-{1-[3-(1H-pyrazol-5-yl)phenyl]piperidin-4-yl}piperidine-3-carboxamide
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
(3aS,6aS)-2-methyl-5-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-6-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2-phenylethyl)-7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,2-dimethyl-1,6-naphthyridine-3-carboxamide
N-methyl-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
N-[(3R,4S)-1-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
(4aR,8aR)-2-(3,5-dichloropyridin-2-yl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
2-[(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)methyl]quinolin-4-ol
4-(3-fluorophenoxy)-1-[2-(pyrrolidin-1-yl)acetyl]piperidine-4-carboxylic acid
2,4-dichloro-3-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenol
(2S)-1-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(2S)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-methyl-2-(propan-2-yl)piperazine
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(pyrrolidin-1-yl)butan-1-one
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-(2-methylphenoxy)ethan-1-one
4-(hydroxymethyl)-1-[3-(pyrrolidine-1-sulfonyl)thiophene-2-carbonyl]piperidin-4-ol
2-amino-4-(4-methanesulfonylphenyl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-5-methyl-1,3-oxazole-4-carboxamide
(4aS,7aR)-1-[(2,5-dimethoxyphenyl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)ethan-1-one
N-[3-(3-chlorophenyl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
2-[(4-amino-6-{[2-(thiophen-2-yl)ethyl]amino}pyrimidin-2-yl)sulfanyl]-N,N-dimethylacetamide
3-{5-[(4-methyl-1,3-thiazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-methyl-4-({methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amino}methyl)benzene-1-sulfonamide
2-(2,3-difluorophenyl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(thian-4-yl)piperazine
N-(2-oxopiperidin-3-yl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[1-(hydroxymethyl)cyclopropanecarbonyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1,4-diazepan-6-ol
1-[(3,4-dimethoxyphenyl)methyl]-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
6-cyclopentyl-1-methyl-N-(2,2,2-trifluoroethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-2-phenylethan-1-one
N2,N2,5,6-tetramethyl-N4-(morpholin-2-ylmethyl)pyrimidine-2,4-diamine
N-(1-methoxypropan-2-yl)-2-methyl-3-[(pyridin-2-ylmethyl)amino]benzamide
5-acetyl-2,4-dimethyl-N-[(3R,5S)-1-(3-methylbut-2-en-1-yl)-5-(methylcarbamoyl)pyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
(1R,2S,9R)-11-(1-benzofuran-2-ylmethyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
3-(3-acetylphenyl)-1-(3-methylbut-2-en-1-yl)-6-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-[(3R,4S)-1-(6-chloro-2-methylquinoline-4-carbonyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-ethyl-2-methylpyrimidin-4-amine
3-(oxan-4-yl)-5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[(3-methylpyridin-4-yl)methyl]benzamide
2-[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
1-[2-(3-chlorophenyl)ethyl]-N-[(1-ethylpyrrolidin-2-yl)methyl]-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(2-fluorophenyl)-3-[(2-phenylethyl)amino]propanamide