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methyl 3-[2-amino-3-cyano-6-(4-hydroxyphenyl)pyridin-4-yl]benzoate
3-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-1-[4-(propylsulfanyl)phenyl]urea
4-[3-(2-methoxyphenoxy)azetidin-1-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
1-[2-(piperazin-1-yl)ethyl]-N-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-(4,7-dimethylquinazolin-2-yl)-N-(5-hydroxyadamantan-2-yl)piperidine-3-carboxamide
3-hydroxy-1-(2-methoxyethyl)-3-[(3-phenoxyazetidin-1-yl)methyl]piperidin-2-one
3-[5-(ethanesulfonyl)thiophen-2-yl]pyridine
4-{[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]methyl}-1-phenylpyrrolidin-2-one
1'-(5-ethyl-1,3,4-oxadiazol-2-yl)spiro[indene-1,4'-piperidine]
2-[3-(dimethylamino)propyl]-9-(6-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
(2R,3R,6R)-5-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4,6-dimethyl-N-{1-oxaspiro[4.4]nonan-3-yl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(phenylamino)pyrimidine-5-carboxamide
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-(3,4,5-trimethoxyphenyl)acetamide
4-(2,3-dihydro-1H-inden-2-yl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({1-[(3,5-dichlorophenyl)methyl]piperidin-3-yl}methyl)-2-hydroxyacetamide
N-(3-chloro-4-methoxyphenyl)-3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}propanamide
5-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
3-(5-chloro-2-methoxybenzoyl)-1-methylpiperidine
3-{2-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}azepan-2-one
N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
1-(2-methylpropyl)-4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-2,4-dimethoxybenzamide
2,6-dimethyl-3-[4-(thian-4-yl)piperazine-1-carbonyl]quinoline
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[4-(pyrimidin-5-yl)-1H-pyrazol-1-yl]acetamide
2-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-3-yl}-4-methyl-1H-1,3-benzodiazole
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)amine
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]acetamide
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
5-[2-(3,4-dimethylpiperazin-1-yl)pyrimidin-4-yl]-2-ethoxybenzoic acid
methyl 2-{4-[2-amino-3-cyano-6-(furan-2-yl)pyridin-4-yl]-2-methoxyphenoxy}acetate
(1S,5R)-3-[2-(2H-1,3-benzodioxol-5-yloxy)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[4-(4-aminoquinazolin-6-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-{[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}-1-(2-methylpropyl)-1H-1,3-benzodiazole
N-[(1s,4s)-4-aminocyclohexyl]-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(prop-2-ene-1-sulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(1-cyclohexyl-1H-pyrazol-5-yl)-3-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]urea
(2R)-2-amino-N-(2,3-dihydro-1H-inden-2-yl)-N,4-dimethylpentanamide
methyl 3-benzamido-1-(furan-2-ylmethyl)-5-[(4-hydroxybutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3aR,6aR)-2-(cyclobutylmethyl)-5-(4-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{1-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-(2-methoxyphenyl)-5-(quinolin-7-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
4-(cyclohex-3-en-1-yl)-1-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-1,2,3-triazole
N-(2,2-difluoroethyl)-4-(quinolin-6-yloxy)piperidine-4-carboxamide
N-(2,2-difluoroethyl)-4-[(1,2-oxazol-3-ylmethyl)sulfamoyl]benzamide
4-{3-[(6-cyclopropylpyrimidin-4-yl)amino]propyl}piperazin-2-one
(1S,5R)-6-(5-chlorothiophene-2-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
[1-(2-ethylpyridine-4-carbonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol