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N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(oxane-4-carbonyl)piperidin-4-yl]propanamide
2-{3-[(1-methylpiperidin-4-yl)methyl]-5-(1-phenyl-1H-1,2,3-triazol-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
7-[(2,3-difluorophenyl)methyl]-2-(2,6-dimethylpyrimidine-4-carbonyl)-2,7-diazaspiro[4.5]decane
(2S)-3-methyl-2-({1-[3-(trifluoromethyl)phenyl]propan-2-yl}amino)butan-1-ol
2-(2-methyl-1,3-thiazole-4-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-(2-methoxy-5-{[(oxan-4-yl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
{3-[(2-methylphenyl)methyl]-1-(5-methylthiophene-2-carbonyl)piperidin-3-yl}methanol
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(3-methylbutanoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(pentan-2-yl)-8-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(1H-indol-5-yl)pyridine-3-carbonitrile
N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(morpholin-3-yl)-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-[4-(2-fluorophenoxy)phenyl]-1-(2-hydroxyethyl)piperidine-4-carboxamide
2-[3-(methylsulfanyl)phenyl]-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
(2R,3S,6R)-5-(1H-1,2,3-benzotriazole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(4-hydroxy-3-methoxyphenyl)methyl]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
[(4-fluorophenyl)methyl](prop-2-en-1-yl){[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
1-(4-methylphenyl)-4-[2-(1-propylpiperidin-4-yl)acetyl]piperazin-2-one
1-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-5-oxopyrrolidine-3-carboxylic acid
{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
N-(3,5-dimethylphenyl)-N'-[(1S)-2-hydroxy-1-phenylethyl]propanediamide
N-[(1S)-1-[1-(4-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl]acetamide
1-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-5-(morpholin-4-ylmethyl)-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
2-{1,3-dimethyl-4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-methyl-2-phenyl-N-(pyridin-2-ylmethyl)acetamide
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
4-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-2-(thiophen-2-yl)-1,3-thiazole
2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1-(morpholin-4-yl)ethan-1-one
4-(1H-indol-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-hydroxy-N-[1-(4-methylpyridin-2-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)urea
2-(4-{[methyl(1-methylpyrrolidin-3-yl)amino]methyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
4-{4-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(quinolin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[1-(pyrimidin-2-yl)piperidin-3-yl]-2-(1H-1,2,4-triazol-1-yl)benzamide
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carbonitrile
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-5-propyl-1,2-oxazole-3-carboxamide
N-[2-(2-ethoxyphenyl)ethyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
7,7-dimethyl-2-(2-phenoxyethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
6-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]-9H-purine
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)acetamide
2-[(1S,5R)-6-[(6-methoxy-2H-chromen-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-(1,3-benzothiazol-6-yl)-1-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]urea
N-[2-(dimethylamino)ethyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-methyl-5-[3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-imidazole
7-{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one