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methyl(2-phenoxyethyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
ethyl 2-[N-methyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]acetate
(4aR,7aS)-1-ethyl-4-(2-methyl-4-phenylpyrimidine-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(6-methoxypyrimidin-4-yl)amino]-1λ6-thiane-1,1-dione
N-{4-[2-(pyridin-2-yl)acetamido]phenyl}pentanamide
N-[2-(dimethylamino)ethyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
3-(4-methyl-1,3-thiazol-5-yl)-1-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}propan-1-one
N-cyclopropyl-N-({2-[methyl(thiophen-3-ylmethyl)amino]-7-(methylsulfanyl)quinolin-3-yl}methyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
methyl 3-cyclopropaneamido-6-({methyl[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
N-(3-chloro-4-methoxyphenyl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)propanamide
2-(azepan-1-yl)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]acetamide
4-acetyl-N-[2-(methylsulfamoyl)phenyl]-1,4-diazepane-1-carboxamide
1-(5-chloro-2-methoxyphenyl)-5-[1-(difluoromethyl)-1H-pyrazol-3-yl]-3-methyl-1H-1,2,4-triazole
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-(3-methoxyphenoxy)-3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propan-2-ol
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-3-(1H-1,2,4-triazol-1-yl)propanamide
5-(2H-1,3-benzodioxol-4-ylmethyl)-3-(3-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-(4-hydroxybutan-2-yl)-1-(oxan-4-ylmethyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-[(1R,3R)-3-aminocyclopentyl]-2-oxo-1,2-dihydroquinoline-3-carboxamide
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-[3-(1H-imidazol-1-yl)propyl]pyrrolidin-2-one
2-(ethoxymethyl)-N-[1-(thiophen-3-yl)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[(3-methoxyphenyl)methyl]-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
N-(dimethyl-1H-1,2,4-triazol-3-yl)-1,4-oxazepane-4-carboxamide
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[2-(pyridin-4-ylsulfanyl)acetyl]pyrrolidin-3-yl]urea
1-(2-hydroxyethyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
5-(2,3-dihydro-1H-inden-2-yl)-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-cyclohexyl-N-(1-methyl-1H-pyrazol-4-yl)-3-oxopiperazine-1-carboxamide
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(quinolin-3-ylmethyl)acetamide
1-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
3-(2-phenylethyl)-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[(4-phenyloxan-4-yl)methyl]amine
N-{[5-chloro-2-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(5-ethyl-1,3-oxazole-4-carbonyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N,N-dimethyl-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine-1-sulfonamide
N-[1-(pyrazin-2-yl)propan-2-yl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-cyclobutyl-5-{1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-[(3S,4R)-1-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-4-propylpyrrolidin-3-yl]acetamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methyl-1H-pyrrole-2-carboxamide
(1S,5R)-6-benzyl-3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]propan-1-one
(1S,5R)-3-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(2-methoxyacetamido)-N,1-dimethyl-N-[2-(oxan-2-yl)ethyl]-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
(3aR,6aR)-2-(2-hydroxyethyl)-5-[(propan-2-yl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(5,6,7-trimethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidine-4-carboxamide
1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(1H-imidazol-2-yl)piperidine