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2-{[(3-chloro-5-fluoro-4-methoxyphenyl)methyl](pyridin-2-ylmethyl)amino}butan-1-ol
3-(2-hydroxyphenyl)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[1-({[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-(2-methoxyphenyl)propanamide
2,6-dimethyl-3-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]quinoline
2-(dimethylamino)-7-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperazine-1-carboxamide
N-(3-hydroxy-3-methylbutyl)-N,1-dimethyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carboxamide
3-[3-(4-fluorophenyl)oxolan-3-yl]-5-(1H-pyrazol-4-yl)-1,2,4-oxadiazole
{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}(methyl)amine
1-[(6-chloropyridin-3-yl)methyl]-4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazine
1-methyl-4-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}-1,4-diazepane
{1-[2-(trifluoromethoxy)benzenesulfonyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
2-({4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}methyl)-6-methylquinolin-4-ol
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]piperidine
2-[(4-methoxyphenyl)amino]-2-methyl-1-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}propan-1-one
2-{5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-(1-ethylpiperidin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]acetamide
3-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
4-[6-amino-5-cyano-4-(5-hydroxy-2-methoxyphenyl)pyridin-2-yl]benzoic acid
2-[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
1-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}-4-(hydroxymethyl)piperidin-4-ol
8-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(2-methylphenyl)methyl]-4-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]piperazine
1-cyclobutanecarbonyl-N-(3-hydroxy-3-phenylpropyl)-N-methylpiperidine-4-carboxamide
3-hydroxy-S-{2-[(3E)-pent-3-enoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}butane-1-sulfonamido
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}propan-1-one
5-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperazine-1-sulfonamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-6-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide
methyl 1-{3-[(3-chlorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
5-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]pyrrolidin-2-yl}-N-propylthiophene-2-carboxamide
ethyl 1-(oxane-4-carbonyl)-4-(2-phenylethyl)piperidine-4-carboxylate
1-{1-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]azetidin-3-yl}-1H-pyrazole
7-(cyclobutylmethyl)-2-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane
(3S,4S)-4-(3-methoxyphenyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-ol
methyl (2S,4R)-1-{[4-(acetyloxy)-3,5-dimethylphenyl]methyl}-4-hydroxypyrrolidine-2-carboxylate
1-methyl-4-phenyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
1-[(1S,5R)-6-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-{5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
6-[(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)amino]pyridine-3-carboxamide
ethyl 4-(1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
methyl 4-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pentanoate
3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-1-methylurea
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5-phenyl-1,2-oxazole-3-carboxamide
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pent-2-yn-1-yl)piperidine
N-[1-(1H-indol-2-yl)ethyl]-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
methyl 2-{5-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetate
N-(2-methoxyethyl)-3,4,7-trimethyl-N-(2-phenoxyethyl)-1H-indole-2-carboxamide