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4-(4-methylphenyl)-N-[(5-methylpyrazin-2-yl)methyl]-5-(pyrimidin-5-yl)pyrimidin-2-amine
4-{5-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
(3S,4S)-1-(2,8-dimethylquinoline-4-carbonyl)-4-(piperidin-1-yl)pyrrolidin-3-ol
N-[(2S)-1-hydroxybutan-2-yl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
3-{[4-(5-ethylfuran-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1,5-dimethyl-1H-indazole
{1-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-3-propylpiperidin-3-yl}methanol
N-cyclopropyl-1-[1-(3-phenylbutyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-(4-acetylphenyl)-3-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}urea
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
3-(2-fluorophenyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidine
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-methyl-6-[3-(methylsulfanyl)propyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetamide
4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[5-(4-methylphenyl)furan-2-yl]formamido}acetic acid
3-{2-tert-butylimidazo[1,2-a]pyrimidin-3-yl}phenol
(2R,6S)-2,6-dimethyl-4-[1-methyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]morpholine
N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyrazine-2-carboxamide
7-fluoro-2-methyl-4-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]quinoline
2-(5-acetylthiophen-3-yl)-1-[2-(4-fluorophenyl)piperidin-1-yl]ethan-1-one
1,5-dimethyl-4-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(4aS,7aR)-1-(1-methylcyclopropanecarbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{[methyl(2-phenylethyl)amino]methyl}-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-4-(pyridin-4-yl)piperazine-1-carboxamide
6-[(pyrimidin-4-ylmethyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
3-[(5,8-dimethoxy-4-methylquinolin-2-yl)amino]-1-methylpyrrolidin-2-one
1-(1-benzylpiperidin-4-yl)-N-propylpiperidine-3-carboxamide
N-[2-(2-chlorophenoxy)ethyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-6-methoxyhexan-1-one
5-tert-butyl-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-1,3,4-oxadiazol-2-amine
1-(3-{[(thian-4-yl)amino]methyl}pyridin-2-yl)piperidin-3-ol
2-(dimethyl-1,3-thiazol-5-yl)-N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
N2-(5,6-dimethylpyrimidin-4-yl)-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
5-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-3-[2-(4-methoxyphenyl)ethyl]-5-methylimidazolidine-2,4-dione
(3S,9aR)-8-(4-chlorobenzoyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
N-cyclopentyl-1-[1-(2-methylpropyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
3-{3-[benzyl(methyl)amino]piperidine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
N-[2-(oxan-3-yl)ethyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2S,4S)-4-amino-1-[2-(morpholin-4-yl)-2-oxoacetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-methyl-8-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-methyl-4-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethoxy}-1,2,5-oxadiazole
6-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-(cyclopropylmethyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-(2-{[4-(methoxycarbonyl)piperazin-1-yl]methyl}phenoxy)acetic acid
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]-1H-indole-6-carboxamide
{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidin-3-yl}methanol
2-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}-1-ethyl-1H-1,3-benzodiazole
methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)[1-(thiophen-2-yl)ethyl]amine
1-{2-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one