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5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)pyrrolidin-2-one
5-[1-(4-fluorobenzoyl)piperidin-4-yl]-3-[(4-fluorophenyl)methyl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
9-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-yl]ethan-1-ol
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-N-(3,4-dimethylphenyl)piperidine-1-carboxamide
1-[2-(4-fluorophenyl)morpholine-4-carbonyl]cyclopropane-1-carboxamide
1-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
4-fluoro-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
2-(1H-indazol-3-yl)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]ethan-1-one
3-[2-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl]pyridine
5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-1-cyclohexyl-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(1R,5R)-N,N-dimethyl-6-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-(3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-4H-1,2,4-triazole
4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-3-methyl-1-propyl-1H-pyrazole
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1,3-thiazole-4-carbonyl)piperidine
8-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-ethyl-2,3-dimethyl-N-(oxan-3-yl)pyrazolo[1,5-a]pyrimidin-7-amine
[(2-fluorophenyl)methyl](2-methoxyethyl){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
1-(3-methoxyphenyl)-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-3-(4-hydroxyphenyl)-2-phenylpropan-1-one
4-(3-methyl-1H-1,2,4-triazol-5-yl)-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine
7-methyl-2-[3-(pyridin-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamido]-N-phenylpropanamide
1-({3-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
1-[(3-fluorophenyl)methyl]-4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
(1S,5R)-6-[(3-chloro-4-methoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(thiophen-2-yl)propan-1-one
1-(2-methoxyethyl)-3-(2-methylpropyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-4H-chromen-4-one
1-ethyl-5-[5-(4-methylphenyl)furan-2-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
methyl 3-(2-methoxy-2-phenylacetyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1R,5R)-3-cyclobutanecarbonyl-6-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-3,5-dimethylfuran-2-carboxamide
ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
3-(3-methoxybenzoyl)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-methylbutanamide
1-[7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-[2-(2-hydroxyethoxy)ethyl]-4-(piperidin-3-yl)benzamide
(1R,2S,4R)-N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
1-({1-[(6-methoxynaphthalen-2-yl)methyl]piperidin-3-yl}methyl)-4-methylpiperazine
3-{[(4aS,7aR)-6,6-dioxo-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
1-ethyl-8-methyl-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-({2-[2-(dimethylamino)ethoxy]phenyl}methyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
N-{2-[2-(propan-2-yloxy)phenyl]ethyl}piperidin-3-amine
4-(4-{1-[1-(1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
1-{3-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]phenyl}ethan-1-one